SCHEMBL3436832

SCHEMBL3436832

COC(C)CN(C)C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13362157 1.00
SCHEMBL12210637 1.00
SCHEMBL20936587 0.81 PIK3CD (0.39)
SCHEMBL18502238 0.78 PIK3CD (0.35)
SCHEMBL2459380 0.78 MAPK1 (0.40)
SCHEMBL20614502 0.78
SCHEMBL21030405 0.77 PIK3CD (0.31)
SCHEMBL22004686 0.77
SCHEMBL19823683 0.77 PIK3CD (0.31)
SCHEMBL12836471 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240229063-A1 TRANSGENIC CORN EVENT ZM_CSM63715 AND METHODS FOR DETECTION AND USES THEREOF MONSANTO TECHNOLOGY LLC (US) 2024-07-11 US disclosed
US-20240025862-A1 SUBSTITUTED N-PHENYLURACILS AND SALTS THEREOF, AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2024-01-25 US disclosed
EP-4230621-A1 SUBSTITUTED N-BENZOIC ACID URACILS, THEIR SALTS AND USE OF SAID COMPOUNDS AS HERBICIDAL AGENTS Bayer AG (DE) 2023-08-23 EP disclosed
EP-4015520-A1 OXYGEN-CONTAINING HETEROCYCLIC COMPOUND, PREPARATION METHOD AND APPLICATION THEREOF Shanghai Yingli Pharmaceutical Co. Ltd. (CN) 2022-06-22 EP disclosed
WO-2022087375-A1 NOVEL HETEROCYCLIC COMPOUNDS SPECTRUM PHARMACEUTICALS, INC. (US) 2022-04-28 WO disclosed
WO-2022002102-A1 QUINAZOLINE COMPOUNDS, PREPARATION METHODS AND USES THEREOF InventisBio Co., Ltd. (CN) 2022-01-06 WO disclosed
WO-2021109737-A1 OXYGEN-CONTAINING HETEROCYCLIC COMPOUND, PREPARATION METHOD AND APPLICATION THEREOF 上海璎黎药业有限公司 2021-06-10 WO disclosed
WO-2021060395-A1 SUSTAINED-RELEASE PHARMACEUTICAL COMPOSITION 持田製薬株式会社 2021-04-01 WO disclosed
WO-2021013800-A1 SUBSTITUTED N-PHENYL-N-AMINOUARCILS AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2021-01-28 WO disclosed
EP-3736277-A1 SUBSTITUTED THIAZOLO-PYRIDINE COMPOUNDS AS MALT1 INHIBITORS Lupin Limited (IN) 2020-11-11 EP disclosed
US-7563921-B2 2-cyano-3(halo)alkoxy-benzenesulfonamide compounds for combating animal pests BASF AKTIENGESELLSCHAFT (DE) 2009-07-21 US disclosed
US-7563921-B2 2-cyano-3(halo)alkoxy-benzenesulfonamide compounds for combating animal pests BASF AKTIENGESELLSCHAFT (DE) 2009-07-21 US disclosed
US-7544637-B2 2-cyano-3(halo)alkoxy-benzenesulfonamide compounds for combating animal pests BASF AKTIENGESELLSCHAFT (DE) 2009-06-09 US disclosed
US-7544637-B2 2-cyano-3(halo)alkoxy-benzenesulfonamide compounds for combating animal pests BASF AKTIENGESELLSCHAFT (DE) 2009-06-09 US disclosed
EP-2009005-A1 AZOLECARBOXAMIDE DERIVATIVE Astellas Pharma Inc. (JP) 2008-12-31 EP disclosed
US-20080306297-A1 NOVEL 2-CYANO-3(HALO)ALKOXY-BENZENESULFONAMIDE COMPOUNDS FOR COMBATING ANIMAL PESTS BASF SE (DE) 2008-12-11 US disclosed
US-20080306297-A1 NOVEL 2-CYANO-3(HALO)ALKOXY-BENZENESULFONAMIDE COMPOUNDS FOR COMBATING ANIMAL PESTS BASF SE (DE) 2008-12-11 US disclosed
US-20080063678-A1 Novel 2-Cyano-3(Halo)Alkoxy-Benzenesulfonamide Compounds for Combating Animal Pests BASF AKTIENGESELLSCHAFT (DE) 2008-03-13 US disclosed
US-20080063678-A1 Novel 2-Cyano-3(Halo)Alkoxy-Benzenesulfonamide Compounds for Combating Animal Pests BASF AKTIENGESELLSCHAFT (DE) 2008-03-13 US disclosed
JP-2005012069-A ELECTROLYTE FOR DRIVING ELECTROLYTIC CAPACITOR NICHICON CORP 2005-01-13 JP disclosed