Evogliptin

Evogliptin

SCHEMBL343846

CC(C)(C)OC[C@@H]1C(=O)NCCN1C(=O)C[C@H](N)Cc1cc(F)c(F)cc1F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DPP4

The experimentally established mechanism targets of Evogliptin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DPP4 known ✓ P27487 19/20 1.00
KCNH2 Q12809 1/20 1.00
DPP8 Q6V1X1 6/20 0.68
DPP7 Q9UHL4 6/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Evogliptin SCHEMBL30866226 1.00 DPP4 (1.00) DPP4KCNH2DPP8DPP7
Evogliptin SCHEMBL18331680 1.00 DPP4 (1.00) DPP4KCNH2DPP8DPP7
Evogliptin SCHEMBL343847 1.00 DPP4 (1.00) DPP4KCNH2DPP8DPP7
Evogliptin SCHEMBL2298513 1.00 DPP4 (1.00) DPP4KCNH2DPP8DPP7
Evogliptin SCHEMBL2496606 0.99 DPP4 (0.98) DPP4KCNH2DPP8DPP7
Evogliptin SCHEMBL2491978 0.99 DPP4 (0.98) DPP4KCNH2DPP8DPP7
Evogliptin SCHEMBL2491981 0.99 DPP4 (0.98) DPP4KCNH2DPP8DPP7
Evogliptin SCHEMBL2493817 0.98 DPP4 (0.96) DPP4KCNH2DPP8DPP7
Evogliptin SCHEMBL2493812 0.98 DPP4 (0.96) DPP4KCNH2DPP8DPP7
Evogliptin SCHEMBL2493525 0.96 DPP4 (0.93) DPP4KCNH2DPP8DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 867 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12636284-B2 Compositions for use in the prevention and/or treatment of intellectual disability and neurodegenerative diseases in a subject with down syndrome Universita' Degli Studi Di Roma “La Sapienza” (IT) 2026-05-26 US claimed
EP-4734978-A2 COMBINATION THERAPIES USING PSILOCYBIN University of Padova (IT) 2026-05-06 EP claimed
EP-4735023-A2 COMPOSITIONS AND METHODS FOR TREATING INFLAMMATORY BOWEL DISEASE Piton Therapeutics, Inc. (US) 2026-05-06 EP claimed
US-12599564-B2 Antidiabetic pharmaceutical compositions Elite Pharmaceutical Solution Inc. (US) 2026-04-14 US claimed
EP-4694979-A2 COMPOUNDS FOR UPREGULATING UTROPHIN LEVELS IN MUSCLE CELLS AND METHOD OF APPLICATION THEREOF Peptris Technologies Private Limited (IN) 2026-02-18 EP claimed
EP-4686474-A1 DPP-IV INHIBITORS FOR THE TREATMENT OR PREVENTION OF AUTOIMMUNE LIVER DISEASES Delta 4 GmbH (AT) 2026-02-04 EP claimed
EP-4596044-A2 COMBINATION THERAPY OF GPR119 AGONISTS AND DPP-4 INHIBITORS Mankind Pharma Ltd. (IN) 2025-08-06 EP claimed
WO-2025104674-A1 COMBINATION THERAPY FOR TREATING NEURODEGENERATIVE DISORDERS ARIBIO CO., LTD. (KR) 2025-05-22 WO claimed
EP-4554574-A2 SMALL MOLECULE REGULATORS OF ALVEOLAR TYPE 2 CELL PROLIFERATION FOR THE TREATMENT OF PULMONARY DISEASES The Scripps Research Institute (US) 2025-05-21 EP claimed
WO-2025100968-A1 USE OF COMPOSITION FOR PREVENTING, ALLEVIATING OR TREATING DIABETIC KIDNEY DISEASE COMPRISING ZINC SALT AND CYCLO-HISPRO AS ACTIVE INGREDIENTS 주식회사 노브메타파마 2025-05-15 WO claimed
EP-3967302-A1 COMPOSITION FOR PREVENTING OR TREATING LIVER DISEASES Acebiomed, Inc. (KR) 2022-03-16 EP claimed
EP-3946343-A1 LOW-DOSE TRIPLE COMBINATION FORMULATION The George Institute For Global Health (AU) 2022-02-09 EP claimed
CN-105555275-B Composition for preventing and treating kidney diseases containing DPP-IV inhibitor 东亚ST株式会社 2021-04-20 CN claimed
EP-2351567-B1 PHARMACEUTICAL COMPOSITION FOR PREVENTION AND TREATMENT OF DIABETES OR OBESITY COMPRISING A COMPOUND THAT INHIBITS ACTIVITY OF DIPEPTIDYL PEPTIDASE-IV, AND OTHER ANTIDIABETIC OR ANTIOBESITY AGENTS AS ACTIVE INGREDIENTS DONG A ST CO LTD (KR) 2017-11-22 EP claimed
EP-2142519-B1 DPP-IV INHIBITOR INCLUDING BETA-AMINO GROUP, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME FOR PREVENTING AND TREATING A DIABETES OR AN OBESITY DONG A PHARM CO LTD (KR) 2014-09-24 EP claimed
US-8440669-B2 Pharmaceutical composition for prevention and treatment of diabetes or obesity comprising a compound that inhibits activity of dipeptidyl peptidase-IV, and other antidiabetic or antiobesity agents as active ingredients DONG-A PHARMACEUTICAL CO. LTD. (KR) 2013-05-14 US claimed
US-8030315-B2 DPP-IV inhibitor including beta-amino group, preparation method thereof and pharmaceutical composition containing the same for preventing and treating diabetes or obesity DONG-A PHARM. CO., LTD. (KR) 2011-10-04 US claimed
US-20110201624-A1 Pharmaceutical Composition for Prevention and Treatment of Diabetes or Obesity Comprising a Compound that Inhibits Activity of Dipeptidyl Peptidase-IV, and other Antidiabetic or Antiobesity Agents as Active Ingredients DONG-A PHARMACEUTICAL. CO., LTD (KR) 2011-08-18 US claimed
EP-2351567-A2 PHARMACEUTICAL COMPOSITION FOR PREVENTION AND TREATMENT OF DIABETES OR OBESITY COMPRISING A COMPOUND THAT INHIBITS ACTIVITY OF DIPEPTIDYL PEPTIDASE-IV, AND OTHER ANTIDIABETIC OR ANTIOBESITY AGENTS AS ACTIVE INGREDIENTS Dong-A Pharmaceutical Co., Ltd. (KR) 2011-08-03 EP claimed
US-20100120790-A1 DPP-IV INHIBITOR INCLUDING BETA-AMINO GROUP, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME FOR PREVENTING AND TREATING DIABETES OR OBESITY DONG-A PHARM. CO., LTD (KR) 2010-05-13 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100120790-A1 DPP-IV INHIBITOR INCLUDING BETA-AMINO GROUP, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME FOR PREVENTING AND TREATING DIABETES OR OBESITY DPP4, DPP7, DPP3 DPP4 1/4885KCNH2 1962/4885DPP8 5/4885
US-12636284-B2 Compositions for use in the prevention and/or treatment of intellectual disability and neurodegenerative diseases in a subject with down syndrome DPP4, DPP3, DPP7 DPP4 1/4885KCNH2 3480/4885DPP8 5/4885
US-12599564-B2 Antidiabetic pharmaceutical compositions GLP1R, DPP4, SLC5A2 DPP4 2/4885KCNH2 1478/4885DPP8 11/4885
US-20110201624-A1 Pharmaceutical Composition for Prevention and Treatment of Diabetes or Obesity Comprising a Compound that Inhibits Activity of Dipeptidyl Peptidase-IV, and other Antidiabetic or Antiobesity Agents as Active Ingredients DPP4, DPP3, DPP7 DPP4 1/4885KCNH2 3038/4885DPP8 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.