SCHEMBL3445474

SCHEMBL3445474

CC(O)CNc1nc(Nc2ccc(Cl)c(C(=O)O)c2)c2nnn(C(C)C)c2n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 6/20 0.52
CDK5 Q00535 4/20 0.52
CDK5R1 Q15078 4/20 0.52
FLT3 P36888 5/20 0.45
CDK2 P24941 2/20 0.44
CCNB1 P14635 2/20 0.44
KDM4E B2RXH2 2/20 0.44
CCNB2 O95067 1/20 0.44
CCNE2 O96020 1/20 0.44
ALDH1A1 P00352 1/20 0.44
NTRK1 P04629 1/20 0.44
INSR P06213 1/20 0.44
PRKACA P17612 1/20 0.44
CCNA2 P20248 1/20 0.44
PRKACG P22612 1/20 0.44
PRKACB P22694 1/20 0.44
CCNE1 P24864 1/20 0.44
MAPK3 P27361 1/20 0.44
CCNA1 P78396 1/20 0.44
NTRK2 Q16620 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3444544 0.93 CDK1 (0.52) CDK1CDK5CDK5R1FLT3CDK2
SCHEMBL3446795 0.92 CDK1 (0.51) CDK1CDK5CDK5R1FLT3CDK2
SCHEMBL3446241 0.90 CDK1 (0.51) CDK1CDK5CDK5R1FLT3CDK2
SCHEMBL3446187 0.90 CDK1 (0.53) CDK1CDK5CDK5R1FLT3CDK2
SCHEMBL3445386 0.89 CDK1 (0.49) CDK1CDK5CDK5R1FLT3CDK2
SCHEMBL3444468 0.86 FLT3 (0.47) CDK1CDK5CDK5R1FLT3CDK2
SCHEMBL3445268 0.85 CDK1 (0.51) CDK1CDK5CDK5R1FLT3CDK2
SCHEMBL3445890 0.84 FLT3 (0.47) CDK1CDK5CDK5R1FLT3CDK2
SCHEMBL3446342 0.84 CDK5 (0.73) CDK1CDK5CDK5R1CDK2CCNB1
SCHEMBL3446334 0.84 CDK5 (0.73) CDK1CDK5CDK5R1CDK2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed