SCHEMBL3445648

SCHEMBL3445648

CC(C)n1nnc2c(Nc3cc(N)cc(Cl)c3)nc(NC3CCC(N)CC3)nc21

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 4/20 0.56
CLK1 P49759 9/20 0.54
CLK2 P49760 9/20 0.54
CLK4 Q9HAZ1 9/20 0.54
CCNB1 P14635 1/20 0.52
CLK3 P49761 1/20 0.52
PDGFRA P16234 6/20 0.51
CCNE1 P24864 6/20 0.51
CDK2 P24941 6/20 0.51
PRKCA P17252 1/20 0.50
FLT3 P36888 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3445788 0.89 CDK1 (0.72) CDK1CLK1CLK2CLK4CCNB1
SCHEMBL3453489 0.89 CDK1 (0.72) CDK1CLK1CLK2CLK4CCNB1
SCHEMBL3445218 0.89 CDK2 (0.62) CDK1PDGFRACCNE1CDK2PRKCA
SCHEMBL3444428 0.87 CDK1 (0.52) CDK1CLK1CLK2CLK4CCNB1
SCHEMBL3444440 0.86 CDK1 (0.54) CDK1PDGFRACCNE1CDK2PRKCA
SCHEMBL3445283 0.86 CDK1 (0.54) CDK1PDGFRACCNE1CDK2PRKCA
SCHEMBL3444351 0.85 CLK1 (0.72) CDK1CLK1CLK2CLK4CCNB1
SCHEMBL3445258 0.85 CDK1 (0.56) CDK1CLK1CLK2CLK4PDGFRA
SCHEMBL3446815 0.84 CDK2 (0.61) CDK1PDGFRACCNE1CDK2PRKCA
SCHEMBL3444543 0.83 FLT3 (0.70) CDK1PDGFRACCNE1CDK2FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed