SCHEMBL3445703

SCHEMBL3445703

CC(N)CNc1nc(NCc2ccccc2)c2nnn(C(C)C)c2n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 10/20 0.60
CCNE1 P24864 7/20 0.60
CCNE2 O96020 6/20 0.60
CCNA2 P20248 5/20 0.60
CCNA1 P78396 5/20 0.60
TDP1 Q9NUW8 3/20 0.55
KDM4E B2RXH2 2/20 0.55
MAPT P10636 2/20 0.55
NPC1 O15118 1/20 0.55
CDK1 P06493 14/20 0.53
CDK5 Q00535 10/20 0.51
CSNK1D P48730 1/20 0.48
CLK2 P49760 1/20 0.48
DYRK1A Q13627 1/20 0.48
HIPK4 Q8NE63 1/20 0.48
SRPK1 Q96SB4 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
CCNB2 O95067 2/20 0.47
CCNB1 P14635 2/20 0.47
CCNB3 Q8WWL7 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3446716 0.89 CDK2 (0.67) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3445042 0.88 CDK2 (0.58) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3446104 0.86 CDK2 (0.51) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3445762 0.86 CDK2 (0.56) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3446162 0.86 CCNE2 (0.46) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3445582 0.83 BCDIN3D (0.50) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3445038 0.83 CDK1 (0.68) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3445903 0.82 CDK2 (0.43) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3445486 0.82 CYP3A4 (0.54) TDP1KDM4EMAPTNPC1CDK1
SCHEMBL3446446 0.81 CDK2 (0.43) CDK2CCNE1CCNE2CCNA2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed