SCHEMBL3445975

SCHEMBL3445975

CCn1nnc2c(Nc3cccc(Cl)c3)nc(NC3CCC(N)CC3)nc21

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 11/20 0.72
PRKCA P17252 3/20 0.72
CCNE1 P24864 8/20 0.65
CDK2 P24941 8/20 0.65
PDGFRA P16234 7/20 0.65
EGFR P00533 2/20 0.58
PAK4 O96013 1/20 0.54
CLK1 P49759 3/20 0.53
CLK2 P49760 3/20 0.53
CCNB1 P14635 2/20 0.53
CLK4 Q9HAZ1 2/20 0.53
NPC1 O15118 1/20 0.53
CCNT1 O60563 1/20 0.53
CDK4 P11802 1/20 0.53
EIF2AK2 P19525 1/20 0.53
CCNA2 P20248 1/20 0.53
CCND1 P24385 1/20 0.53
CCND3 P30281 1/20 0.53
MTOR P42345 1/20 0.53
CDK7 P50613 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3445258 0.89 CDK1 (0.56) CDK1PRKCACCNE1CDK2PDGFRA
SCHEMBL3445305 0.89 PDGFRA (0.63) CDK1PRKCACCNE1CDK2PDGFRA
SCHEMBL3445623 0.89 PDGFRA (0.62) CDK1PRKCACCNE1CDK2PDGFRA
SCHEMBL3444708 0.88 CDK1 (0.67) CDK1PRKCACCNE1CDK2PDGFRA
SCHEMBL3445758 0.86 CDK1 (0.54) CDK1PRKCACCNE1CDK2PDGFRA
SCHEMBL3445839 0.86 CDK1 (0.54) CDK1PRKCACCNE1CDK2PDGFRA
SCHEMBL3444766 0.86 CLK1 (0.73) CDK1PRKCACCNE1CDK2EGFR
SCHEMBL3453489 0.85 CDK1 (0.72) CDK1PRKCACCNE1CDK2PDGFRA
SCHEMBL3445788 0.85 CDK1 (0.72) CDK1PRKCACCNE1CDK2PDGFRA
SCHEMBL8707068 0.84 CDK1 (1.00) CDK1PRKCACCNE1CDK2PDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed