SCHEMBL3446702

SCHEMBL3446702

CCC(CO)Nc1nc(Nc2ccc(Cl)cc2)c2nnn(CC)c2n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 15/20 0.52
CDK5R1 Q15078 15/20 0.52
KDM4E B2RXH2 3/20 0.52
MAPT P10636 2/20 0.52
NPC1 O15118 1/20 0.52
POLB P06746 1/20 0.52
CDK2 P24941 14/20 0.51
CCNA2 P20248 13/20 0.51
CCNA1 P78396 13/20 0.51
DYRK1A Q13627 13/20 0.51
CDK1 P06493 2/20 0.48
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
KMT2A Q03164 1/20 0.48
CCNT1 O60563 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK9 P50750 1/20 0.43
CRHR1 P34998 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3444438 0.90 CDK5 (0.51) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3444633 0.90 CDK5 (0.52) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3446707 0.89 CDK5 (0.52) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3445426 0.88 CDK5 (0.67) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3444447 0.87 CDK1 (0.65) CDK5CDK5R1KDM4EMAPTCDK2
SCHEMBL3444445 0.87 CDK1 (0.65) CDK5CDK5R1KDM4EMAPTCDK2
SCHEMBL3444971 0.87 CDK5 (0.55) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3445024 0.87 CDK5 (0.49) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3446747 0.87 CDK5 (0.49) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3444618 0.86 CDK1 (0.51) CDK5CDK5R1KDM4EMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed