Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL3459082

C[C@@H](Cc1cccs1)Nc1cc[nH]c(=O)c1-c1nc2cc3c(cc2[nH]1)CN(CCCN1CCCC1)C3=O.O=C(O)C(F)(F)F

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 12/20 0.55
ACVRL1 P37023 12/20 0.55
RET P07949 5/20 0.55
ROS1 P08922 5/20 0.55
NTRK3 Q16288 2/20 0.55
NTRK2 Q16620 2/20 0.55
MET P08581 2/20 0.54
HTR4 Q13639 2/20 0.34
IGF1R P08069 5/20 0.33
JAK1 P23458 1/20 0.33
CYP3A4 P08684 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3465417 0.94 NTRK1 (0.59) NTRK1ACVRL1RETROS1NTRK3
SCHEMBL13692318 0.94 NTRK1 (0.59) NTRK1ACVRL1RETROS1NTRK3
SCHEMBL13692266 0.92 NTRK1 (0.55) NTRK1ACVRL1RETROS1NTRK3
SCHEMBL3459663 0.92 NTRK1 (0.55) NTRK1ACVRL1RETROS1NTRK3
SCHEMBL13692264 0.92 NTRK1 (0.55) NTRK1ACVRL1RETROS1NTRK3
SCHEMBL13692530 0.91 NTRK1 (0.55) NTRK1ACVRL1RETROS1NTRK3
SCHEMBL13692361 0.88 NTRK1 (0.56) NTRK1ACVRL1RETROS1NTRK3
Trifluoroacetic Acid SCHEMBL14719368 0.86 NTRK1 (0.56) NTRK1ACVRL1RETROS1NTRK3
Trifluoroacetic Acid SCHEMBL14718959 0.86 NTRK1 (0.55) NTRK1ACVRL1RETROS1NTRK3
Trifluoroacetic Acid SCHEMBL3469072 0.86 NTRK1 (0.55) NTRK1ACVRL1RETROS1NTRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262807-A1 NOVEL TYROSINE KINASE INHIBITORS ChemBridge Corporation (US) 2010-12-22 EP disclosed
WO-2009117097-A1 NOVEL TYROSINE KINASE INHIBITORS CHEMBRIDGE CORPORATION (US) 2009-09-24 WO disclosed