Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | ORAI1 | Q96D31 | 1/20 | 0.48 |
| ▸ | ORAI2 | Q96SN7 | 1/20 | 0.48 |
| ▸ | ORAI3 | Q9BRQ5 | 1/20 | 0.48 |
| ▸ | TRPV6 | Q9H1D0 | 1/20 | 0.48 |
| ▸ | KDM4E | B2RXH2 | 2/20 | 0.42 |
| ▸ | ALDH1A1 | P00352 | 2/20 | 0.42 |
| ▸ | MEN1 | O00255 | 1/20 | 0.42 |
| ▸ | TRPM2 | O94759 | 1/20 | 0.42 |
| ▸ | CYP1A2 | P05177 | 1/20 | 0.42 |
| ▸ | CYP3A4 | P08684 | 1/20 | 0.42 |
| ▸ | THRB | P10828 | 1/20 | 0.42 |
| ▸ | HPGD | P15428 | 1/20 | 0.42 |
| ▸ | ALOX15 | P16050 | 1/20 | 0.42 |
| ▸ | TSHR | P16473 | 1/20 | 0.42 |
| ▸ | ALOX12 | P18054 | 1/20 | 0.42 |
| ▸ | MAPK1 | P28482 | 1/20 | 0.42 |
| ▸ | KMT2A | Q03164 | 1/20 | 0.42 |
| ▸ | TDP1 | Q9NUW8 | 1/20 | 0.42 |
| ▸ | SLC6A2 | P23975 | 2/20 | 0.37 |
| ▸ | TAAR1 | Q96RJ0 | 2/20 | 0.37 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL7461066 | 0.81 | ORAI1 (0.52) | ORAI1ORAI2ORAI3TRPV6KDM4E | |
| SCHEMBL4174754 | 0.78 | KDM4E (0.42) | ORAI1ORAI2ORAI3TRPV6KDM4E | |
| SCHEMBL2407845 | 0.78 | ORAI1 (0.40) | ORAI1ORAI2ORAI3TRPV6KDM4E | |
| SCHEMBL5710601 | 0.72 | ORAI1 (0.48) | ORAI1ORAI2ORAI3TRPV6KDM4E | |
| SCHEMBL12270707 | 0.71 | DPP4 (0.48) | ORAI1ORAI2ORAI3TRPV6KDM4E | |
| SCHEMBL2404970 | 0.70 | CYP3A4 (0.49) | ORAI1ORAI2ORAI3TRPV6KDM4E | |
| SCHEMBL12318751 | 0.70 | ORAI1 (0.40) | ORAI1ORAI2ORAI3TRPV6KDM4E | |
| SCHEMBL2031393 | 0.70 | ANPEP (0.38) | TSHRSLC6A2TAAR1MAOASLC6A4 | |
| SCHEMBL2407157 | 0.70 | IDO1 (0.30) | — | |
| SCHEMBL10454943 | 0.69 | SLC6A2 (0.41) | ORAI1ORAI2ORAI3TRPV6KDM4E |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-3808348-A1 | COMPOSITIONS AND METHODS FOR THE TREATMENT OF PROGRESSIVE MULTIFOCAL LEUKOENCEPHALOPATHY (PML) | Biogen MA Inc. (US) | 2021-04-21 | — | — | EP | claimed |
| US-20130183289-A1 | COMPOSITIONS AND METHODS FOR THE TREATMENT OF PROGRESSIVE MULTIFOCAL LEUKOENCEPHALOPATHY (PML) | BIOGEN IDEC MA INC (US) | 2013-07-18 | — | — | US | claimed |
| EP-2200611-A1 | COMPOSITIONS AND METHODS FOR THE TREATMENT OF PROGRESSIVE MULTIFOCAL LEUKOENCEPHALOPATHY (PML) | Biogen Idec MA, Inc. (US) | 2010-06-30 | — | — | EP | claimed |
| WO-2009038684-A1 | COMPOSITIONS AND METHODS FOR THE TREATMENT OF PROGRESSIVE MULTIFOCAL LEUKOENCEPHALOPATHY (PML) | BIOGEN IDEC MA INC. (US) | 2009-03-26 | — | — | WO | claimed |
| EP-3808348-A1 | COMPOSITIONS AND METHODS FOR THE TREATMENT OF PROGRESSIVE MULTIFOCAL LEUKOENCEPHALOPATHY (PML) | Biogen MA Inc. (US) | 2021-04-21 | — | — | EP | disclosed |
| EP-3025714-B9 | COMPOSITIONS AND METHODS FOR THE TREATMENT OF PROGRESSIVE MULTIFOCAL LEUKOENCEPHALOPATHY (PML) | BIOGEN MA INC (US) | 2020-11-18 | — | — | EP | disclosed |
| EP-3025714-B1 | COMPOSITIONS AND METHODS FOR THE TREATMENT OF PROGRESSIVE MULTIFOCAL LEUKOENCEPHALOPATHY (PML) | BIOGEN MA INC (US) | 2020-07-15 | — | — | EP | disclosed |
| US-20200197544-A1 | JCV IMAGING METHODS AND COMPOSITIONS | BIOGEN MA INC (US) | 2020-06-25 | — | — | US | disclosed |
| EP-3615681-A1 | JCV IMAGING METHODS AND COMPOSITIONS | Biogen MA Inc. (US) | 2020-03-04 | — | — | EP | disclosed |
| EP-2869826-B1 | PEST REPELLENTS FROM PLANT EXTRACTS | EDEN SHIELD LTD (IL) | 2019-05-15 | — | — | EP | disclosed |
| WO-2018200791-A1 | JCV IMAGING METHODS AND COMPOSITIONS | BIOGEN MA INC. (US) | 2018-11-01 | — | — | WO | disclosed |
| EP-2890689-B1 | DIHYDROCHALCONE DERIVATIVES AND THEIR USE AS ANTIBIOTIC AGENTS | UNIV DU QUEBEC A CHICOUTIMI (CA) | 2018-08-08 | — | — | EP | disclosed |
| WO-1999034810-A1 | A PROCESS FOR THE ISOLATION, RECOVERY AND PURIFICATION OF NON-POLAR EXTRACTIVES | HER MAJESTY IN RIGHT OF CANADA AS REPRESENTED BY THE MINISTER OF AGRICULTURE AND AGRI-FOOD CANADA (CA) | 1999-07-15 | — | — | WO | disclosed |
| US-5753697-A | ANTIRADICAL AND-OR ANTILIPOPEROXIDATIVE AND-OR HEPATOTROPIC PROPERTIES | LABORATOIRES DOLISOS (FR) | 1998-05-19 | — | — | US | disclosed |
| WO-1997011951-A1 | FUNGICIDES | ZENECA LIMITED (GB) | 1997-04-03 | — | — | WO | disclosed |
| EP-0449557-B1 | Recovery of values from cereal wastes | CA MINISTER AGRICULTURE & FOOD (CA) | 1996-09-04 | — | — | EP | disclosed |
| EP-0706392-A1 | USE OF ROSMANOL DERIVATIVES FOR PRODUCING ANTIRADICAL AND/OR ANTILIPOPEROXIDATIVE AND/OR HEPATOTROPIC DRUGS | LABORATOIRES DOLISOS (FR) | 1996-04-17 | — | — | EP | disclosed |
| WO-1995001174-A1 | USE OF ROSMANOL DERIVATIVES FOR PRODUCING ANTIRADICAL AND/OR ANTILIPOPEROXIDATIVE AND/OR HEPATOTROPIC DRUGS | LABORATOIRES DOLISOS (FR) | 1995-01-12 | — | — | WO | disclosed |
| US-5169660-A | Steeping cereals in water to liquify endosperm, then macerating them in aqueous ethanol solution, separation and recovery of bran and endosperm materials | HER MAJESTY THE QUEEN IN RIGHT OF CANADA, AS REPRESENTED BY THE MINISTER OF AGRICULTURE (CA) | 1992-12-08 | — | — | US | disclosed |
| EP-0449557-A2 | Recovery of values from cereal wastes | Her Majesty in Right of Canada as represented by the Minister of Agriculture Canada (CA) | 1991-10-02 | — | — | EP | disclosed |