SCHEMBL3466232

SCHEMBL3466232

CC1CCCCN1c1ccc(-c2nc(-c3ccc4[nH]ccc4c3)no2)cc1C#N.CC1CCCCN1c1ccc(-c2nc(-c3ccc4[nH]ccc4c3)no2)cc1NS(C)(=O)=O

nearest known ligand 0.88

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 14/20 0.88
TP53 P04637 2/20 0.44
POLB P06746 1/20 0.41
PIK3CA P42336 2/20 0.39
MTOR P42345 2/20 0.39
S1PR3 Q99500 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2415693 0.94 S1PR1 (1.00) S1PR1TP53POLBPIK3CAMTOR
SCHEMBL2415287 0.90 S1PR1 (0.70) S1PR1TP53POLBS1PR3
SCHEMBL13345821 0.88 S1PR1 (0.88) S1PR1TP53POLBPIK3CAMTOR
SCHEMBL13346042 0.79 S1PR1 (0.73) S1PR1TP53POLBS1PR3
SCHEMBL2410798 0.78 S1PR1 (0.65) S1PR1TP53POLB
SCHEMBL2806750 0.78 S1PR1 (0.71) S1PR1TP53POLB
SCHEMBL2414988 0.77 S1PR1 (1.00) S1PR1TP53POLB
SCHEMBL2773184 0.76 S1PR1 (0.69) S1PR1TP53POLB
SCHEMBL2772257 0.76 S1PR1 (0.69) S1PR1TP53POLB
SCHEMBL2770910 0.76 S1PR1 (0.68) S1PR1TP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010069949-A1 OXADIAZOLE FUSED HETEROCYCLIC DERIVATIVES USEFUL FOR THE TREATMENT OF MULTIPLE SCLEROSIS MERCK SERONO S.A. (CH) 2010-06-24 WO disclosed