SCHEMBL3467029

SCHEMBL3467029

C#Cc1nc(-c2ccc(S(=O)(=O)C(C)C)cc2)cnc1C(=O)N(C(=O)O)C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ATR Q13535 20/20 0.41
ATM Q13315 7/20 0.41
PRKDC P78527 4/20 0.41
GSK3B P49841 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3055887 0.95 ATR (0.41) ATRATMPRKDCGSK3B
SCHEMBL15684385 0.85 ATR (0.44) ATRATMPRKDCGSK3B
SCHEMBL667416 0.84 ATR (0.40) ATRATMPRKDCGSK3B
SCHEMBL667542 0.82 ATR (0.41) ATRATMPRKDCGSK3B
SCHEMBL19102162 0.78 ATR (0.38) ATRATMPRKDCGSK3B
SCHEMBL667206 0.74 ATR (0.39) ATRATMPRKDCGSK3B
SCHEMBL14829434 0.74 ATR (0.42) ATRATMPRKDCGSK3B
SCHEMBL10141979 0.73 ATR (0.41) ATRATMPRKDCGSK3B
SCHEMBL15684386 0.71 ATR (0.43) ATRATMPRKDCGSK3B
SCHEMBL29243957 0.71 ATR (0.45) ATRATMPRKDCGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010071837-A1 PYRAZINE DERIVATIVES USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-06-24 WO disclosed