SCHEMBL3467253

SCHEMBL3467253

COc1cc(C2CCN(CC(=O)NCC(O)CO)CC2)ccc1Nc1ncc2ccc(-c3ccccc3OC)n2n1

nearest known ligand 0.80

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 18/20 0.80
NPM1 P06748 14/20 0.80
INSR P06213 11/20 0.80
JAK2 O60674 3/20 0.77
PTK2 Q05397 2/20 0.77
CYP3A4 P08684 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
KCNH2 Q12809 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL522455 0.90 ALK (0.82) ALKNPM1INSRJAK2PTK2
SCHEMBL519683 0.89 ALK (1.00) ALKNPM1INSRJAK2PTK2
SCHEMBL520989 0.88 ALK (1.00) ALKNPM1INSRJAK2PTK2
SCHEMBL520990 0.88 ALK (1.00) ALKNPM1INSRJAK2PTK2
SCHEMBL521004 0.88 ALK (0.87) ALKNPM1INSRJAK2PTK2
SCHEMBL520841 0.87 ALK (1.00) ALKNPM1INSRJAK2PTK2
SCHEMBL520417 0.86 ALK (0.83) ALKNPM1INSRJAK2PTK2
SCHEMBL16267902 0.84 ALK (0.81) ALKNPM1INSRJAK2PTK2
SCHEMBL522231 0.84 ALK (0.81) ALKNPM1INSRJAK2PTK2
SCHEMBL519543 0.84 ALK (1.00) ALKNPM1INSRJAK2PTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010071885-A1 PYRROLOTRIAZINES AS ALK AND JAK2 INHIBITORS CEPHALON, INC. (US) 2010-06-24 WO disclosed