SCHEMBL3467258

SCHEMBL3467258

COc1ccc(CNC(=O)c2cn(CCCCCC(=O)NO)c3ccccc3c2=O)cc1

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 10/20 0.68
HDAC6 Q9UBN7 9/20 0.68
CHRM1 P11229 1/20 0.52
CNR2 P34972 2/20 0.52
HDAC3 O15379 2/20 0.52
HDAC2 Q92769 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3467496 0.90 HDAC1 (0.73) HDAC1HDAC6CNR2HDAC3HDAC2
SCHEMBL3468139 0.88 CNR2 (0.58) HDAC1HDAC6CNR2HDAC3HDAC2
SCHEMBL3477433 0.88 HDAC1 (0.71) HDAC1HDAC6CNR2HDAC3HDAC2
SCHEMBL3466885 0.81 HDAC6 (0.59) HDAC1HDAC6CNR2HDAC3HDAC2
SCHEMBL7919669 0.81 HDAC1 (0.61) HDAC1HDAC6CNR2HDAC3HDAC2
SCHEMBL3467874 0.79 HDAC6 (0.57) HDAC1HDAC6CNR2HDAC3HDAC2
SCHEMBL7912521 0.79 HDAC3 (0.59) HDAC1HDAC6CNR2HDAC3HDAC2
SCHEMBL7919673 0.79 HDAC1 (0.58) HDAC1HDAC6CNR2
SCHEMBL3467928 0.79 HDAC1 (0.60) HDAC1HDAC6CNR2HDAC3HDAC2
SCHEMBL3467026 0.78 CNR2 (0.51) HDAC1HDAC6CNR2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010073078-A2 HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LTD. (IN) 2010-07-01 WO disclosed