SCHEMBL3468320

SCHEMBL3468320

N#Cc1cnc2ccc(N)cc2c1Nc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 9/20 0.60
EGFR P00533 7/20 0.60
ERBB2 P04626 6/20 0.60
RAF1 P04049 5/20 0.60
MAP3K8 P41279 2/20 0.51
STK4 Q13043 1/20 0.50
PDE4B Q07343 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28769852 0.90 MAP2K1 (0.67) MAP2K1EGFRERBB2RAF1MAP3K8
SCHEMBL15320481 0.90 MAP2K1 (0.77) MAP2K1EGFRERBB2RAF1MAP3K8
SCHEMBL27707326 0.88 EGFR (0.53) MAP2K1EGFRERBB2RAF1MAP3K8
SCHEMBL1893034 0.88 EGFR (0.65) EGFRERBB2MAP3K8PDE4B
SCHEMBL27728172 0.88 EGFR (0.55) MAP2K1EGFRERBB2RAF1MAP3K8
SCHEMBL1897881 0.87 EGFR (0.64) MAP2K1EGFRERBB2RAF1MAP3K8
SCHEMBL1892933 0.87 EGFR (0.60) EGFRERBB2MAP3K8PDE4B
SCHEMBL1893339 0.87 EGFR (0.70) EGFRERBB2
SCHEMBL6381746 0.87 EGFR (0.66) EGFRERBB2MAP3K8PDE4B
SCHEMBL9911596 0.87 EGFR (0.60) EGFRERBB2MAP3K8PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111848581-B Preparation method of 3-cyano-4-anilino-6-aminoquinoline derivative 昆明学院 2021-08-10 CN claimed
CN-111848581-A Preparation method of 3-cyano-4-anilino-6-aminoquinoline derivative 昆明学院 2020-10-30 CN claimed
CN-111848581-B Preparation method of 3-cyano-4-anilino-6-aminoquinoline derivative 昆明学院 2021-08-10 CN disclosed
CN-111848581-B Preparation method of 3-cyano-4-anilino-6-aminoquinoline derivative 昆明学院 2021-08-10 CN disclosed
CN-111848581-B Preparation method of 3-cyano-4-anilino-6-aminoquinoline derivative 昆明学院 2021-08-10 CN disclosed
CN-111848581-A Preparation method of 3-cyano-4-anilino-6-aminoquinoline derivative 昆明学院 2020-10-30 CN disclosed
CN-111848581-A Preparation method of 3-cyano-4-anilino-6-aminoquinoline derivative 昆明学院 2020-10-30 CN disclosed
CN-111848581-A Preparation method of 3-cyano-4-anilino-6-aminoquinoline derivative 昆明学院 2020-10-30 CN disclosed
WO-2010076764-A1 IRREVERSIBLE EGFR INHIBITOR COMPOUNDS WITH ANTIPROLIFERATIVE ACTIVITY UNIVERSITA' DEGLI STUDI DI PARMA (IT) 2010-07-08 WO disclosed