SCHEMBL3468644

SCHEMBL3468644

Cn1c(N2CCNC(c3ccc(N4CCOCC4)cc3)C2)nc(-c2ccncc2F)cc1=O

nearest known ligand 0.63

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 19/20 0.63
CYP2D6 P10635 2/20 0.63
CYP1A2 P05177 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL82511 1.00 GSK3B (0.63) GSK3BCYP2D6CYP1A2
SCHEMBL87855 0.93 GSK3B (0.64) GSK3BCYP2D6CYP1A2
SCHEMBL87886 0.93 GSK3B (0.64) GSK3BCYP2D6CYP1A2
SCHEMBL83720 0.92 GSK3B (0.63) GSK3BCYP2D6CYP1A2
SCHEMBL83029 0.92 GSK3B (0.63) GSK3BCYP2D6CYP1A2
Hydrochloric Acid SCHEMBL83055 0.92 GSK3B (0.62) GSK3BCYP2D6CYP1A2
SCHEMBL87869 0.92 GSK3B (0.64) GSK3BCYP2D6CYP1A2
SCHEMBL87870 0.90 GSK3B (0.60) GSK3BCYP2D6CYP1A2
SCHEMBL87918 0.90 GSK3B (0.60) GSK3BCYP2D6CYP1A2
SCHEMBL87728 0.90 GSK3B (0.59) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2261224-A2 6-(Pyridinyl)-4-pyrimidone derivatives as tau protein kinase 1 inhibitors Mitsubishi Tanabe Pharma Corporation (JP) 2010-12-15 EP disclosed