SCHEMBL3469342

SCHEMBL3469342

O=c1ccc2ncc(F)c3c2n1CC3(O)CN1CCC(NCc2cc3c(cn2)OCS3)CC1

nearest known ligand 0.66

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 14/20 0.66
SLC2A1 P11166 2/20 0.45
TOP2A P11388 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2768409 1.00 KCNH2 (0.66) KCNH2SLC2A1TOP2A
SCHEMBL2768016 1.00 KCNH2 (0.66) KCNH2SLC2A1TOP2A
SCHEMBL2767951 0.94 KCNH2 (0.68) KCNH2SLC2A1TOP2A
SCHEMBL2767542 0.94 KCNH2 (0.68) KCNH2SLC2A1TOP2A
SCHEMBL13244867 0.91 KCNH2 (0.56) KCNH2SLC2A1TOP2A
SCHEMBL3469114 0.91 KCNH2 (0.56) KCNH2SLC2A1TOP2A
SCHEMBL2768460 0.91 KCNH2 (0.54) KCNH2SLC2A1
SCHEMBL3478626 0.91 KCNH2 (0.54) KCNH2SLC2A1
Hydrochloric Acid SCHEMBL2768275 0.90 KCNH2 (0.53) KCNH2SLC2A1
Hydrochloric Acid SCHEMBL2770784 0.90 KCNH2 (0.53) KCNH2SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2167196-A1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS Glaxo Group Limited (GB) 2010-03-31 EP disclosed
WO-2009000745-A1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed