SCHEMBL3469487

SCHEMBL3469487

COc1ccccc1-c1ccc2cnc(Nc3ccc(CN4CCN(C)CC4)cc3)nn12.COc1ccccc1-c1ccc2cnc([S+](C)[O-])nn12

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 14/20 0.64
ALK Q9UM73 7/20 0.64
INSR P06213 4/20 0.64
CYP3A4 P08684 1/20 0.64
NPM1 P06748 3/20 0.53
PTK2 Q05397 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL519705 0.92 JAK2 (0.75) JAK2ALKINSRCYP3A4NPM1
SCHEMBL521546 0.85 JAK2 (0.70) JAK2ALKINSRCYP3A4NPM1
SCHEMBL520022 0.82 JAK2 (0.60) JAK2ALKINSRCYP3A4NPM1
SCHEMBL520790 0.81 ALK (0.73) JAK2ALKINSRCYP3A4NPM1
SCHEMBL522459 0.81 ALK (0.73) JAK2ALKINSRCYP3A4NPM1
SCHEMBL519058 0.80 JAK2 (0.73) JAK2ALKINSRCYP3A4NPM1
SCHEMBL2510881 0.80 JAK2 (0.71) JAK2ALKINSRCYP3A4NPM1
SCHEMBL2521959 0.79 JAK2 (1.00) JAK2ALKINSRCYP3A4NPM1
SCHEMBL519194 0.78 JAK2 (0.55) JAK2ALKINSRCYP3A4NPM1
SCHEMBL520566 0.77 JAK2 (0.81) JAK2ALKINSRCYP3A4NPM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010071885-A1 PYRROLOTRIAZINES AS ALK AND JAK2 INHIBITORS CEPHALON, INC. (US) 2010-06-24 WO disclosed