SCHEMBL3469855

SCHEMBL3469855

C1CN2CC12.CCN1Cc2cc3[nH]c(-c4c(Cl)cc[nH]c4=O)nc3cc2C1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 11/20 0.47
ACVRL1 P37023 11/20 0.47
RET P07949 5/20 0.47
ROS1 P08922 5/20 0.47
NTRK3 Q16288 2/20 0.47
NTRK2 Q16620 2/20 0.47
MET P08581 2/20 0.43
JAK1 P23458 4/20 0.35
HRH4 Q9H3N8 1/20 0.34
IGF1R P08069 2/20 0.34
CYP3A4 P08684 2/20 0.34
PDGFRB P09619 1/20 0.33
FGFR1 P11362 1/20 0.33
KDR P35968 1/20 0.33
NUAK1 O60285 1/20 0.33
JAK2 O60674 1/20 0.33
PDGFRA P16234 1/20 0.33
TYK2 P29597 1/20 0.33
FLT3 P36888 1/20 0.33
JAK3 P52333 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3469078 0.99 NTRK1 (0.47) NTRK1ACVRL1RETROS1NTRK3
SCHEMBL773090 0.81 NTRK1 (0.64) NTRK1ACVRL1RETROS1NTRK3
Hydrochloric Acid SCHEMBL768310 0.81 NTRK1 (0.63) NTRK1ACVRL1RETROS1NTRK3
SCHEMBL3461158 0.80 NTRK1 (0.57) NTRK1ACVRL1RETROS1NTRK3
SCHEMBL768143 0.79 NTRK1 (0.54) NTRK1ACVRL1RETROS1NTRK3
SCHEMBL13692321 0.78 NTRK1 (0.48) NTRK1ACVRL1RETROS1NTRK3
Hydrochloric Acid SCHEMBL768584 0.78 NTRK1 (0.53) NTRK1ACVRL1RETROS1NTRK3
SCHEMBL767789 0.78 NTRK1 (0.59) NTRK1ACVRL1RETROS1NTRK3
Hydrochloric Acid SCHEMBL3466822 0.78 NTRK1 (0.47) NTRK1ACVRL1RETROS1NTRK3
SCHEMBL438635 0.77 NTRK1 (0.60) NTRK1ACVRL1RETROS1NTRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262807-A1 NOVEL TYROSINE KINASE INHIBITORS ChemBridge Corporation (US) 2010-12-22 EP disclosed
WO-2009117097-A1 NOVEL TYROSINE KINASE INHIBITORS CHEMBRIDGE CORPORATION (US) 2009-09-24 WO disclosed