SCHEMBL3474835

SCHEMBL3474835

Clc1c(-c2ccc3c(nnn3CC3CC3)c2Cl)ccnc1N1CCOCC1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 13/20 0.45
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 3/20 0.38
GAA P10253 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ATR Q13535 1/20 0.36
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3475146 0.92 GRM2 (0.42) GRM2ALDH1A1KDM4EGAAL3MBTL1
SCHEMBL3475658 0.90 GRM2 (0.46) GRM2ALDH1A1KDM4EGAAL3MBTL1
SCHEMBL3476720 0.80 CNR2 (0.52) GRM2
SCHEMBL3475327 0.77 GRM2 (0.46) GRM2ALDH1A1KDM4EGAALMNA
SCHEMBL13823754 0.76 NPSR1 (0.46) GRM2
SCHEMBL3476639 0.75 GRM2 (0.54) GRM2
SCHEMBL3474663 0.73 GRM2 (0.42) GRM2
SCHEMBL3475353 0.73 GRM2 (0.42) GRM2KDM4EL3MBTL1
SCHEMBL3476538 0.73 GRM2 (0.52) GRM2
SCHEMBL3476566 0.73 GRM2 (0.52) GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO claimed
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO disclosed
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO disclosed