SCHEMBL3476006

SCHEMBL3476006

Cc1cc(-c2ccc3c(nnn3CC3CC3)c2Cl)ccc1CO

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 14/20 0.46
TDO2 P48775 5/20 0.41
SGK1 O00141 1/20 0.36
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3475409 0.84 GRM2 (0.53) GRM2TDO2MAPK14
SCHEMBL3473877 0.81 GRM2 (0.53) GRM2TDO2
SCHEMBL3475688 0.81 GRM2 (0.49) GRM2TDO2
SCHEMBL3474008 0.81 GRM2 (0.55) GRM2TDO2
SCHEMBL13823853 0.80 GRM2 (0.51) GRM2TDO2
SCHEMBL7816044 0.80 GRM2 (0.53) GRM2TDO2
SCHEMBL3475381 0.80 GRM2 (0.53) GRM2TDO2
SCHEMBL3475089 0.80 GRM2 (0.48) GRM2TDO2
SCHEMBL3477455 0.80 GRM2 (0.48) GRM2TDO2
SCHEMBL7809962 0.80 GRM2 (0.48) GRM2TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO claimed
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO disclosed
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO disclosed