SCHEMBL3476401

SCHEMBL3476401

CC(C)(C)N1CCN(c2ccc(-c3ccc4c(nnn4CC4CC4)c3Cl)cn2)CC1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 10/20 0.41
CNR2 P34972 6/20 0.39
CNR1 P21554 1/20 0.39
AURKA O14965 3/20 0.36
AXL P30530 3/20 0.36
FLT3 P36888 3/20 0.36
RET P07949 3/20 0.35
KIT P10721 2/20 0.35
SRC P12931 2/20 0.35
KDR P35968 2/20 0.35
MERTK Q12866 2/20 0.35
MET P08581 1/20 0.35
PDGFRA P16234 1/20 0.35
TYRO3 Q06418 1/20 0.35
DDR1 Q08345 1/20 0.35
AURKB Q96GD4 1/20 0.35
ALK Q9UM73 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3474286 0.90 RET (0.43) GRM2CNR2CNR1AURKAAXL
SCHEMBL3474262 0.86 GRM2 (0.43) GRM2CNR2CNR1AURKAAXL
SCHEMBL3476720 0.86 CNR2 (0.52) GRM2CNR2CNR1
SCHEMBL3474206 0.85 RET (0.46) RET
SCHEMBL3475599 0.81 GRM2 (0.46) GRM2
SCHEMBL3475688 0.80 GRM2 (0.49) GRM2
SCHEMBL3476498 0.80 GRM2 (0.51) GRM2
SCHEMBL3475824 0.79 GRM2 (0.49) GRM2KDR
SCHEMBL3477455 0.79 GRM2 (0.48) GRM2
SCHEMBL3476219 0.78 GRM2 (0.49) GRM2CNR2AXLMERTKTYRO3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO claimed