SCHEMBL3476922

SCHEMBL3476922

CC(C)(O)c1cncc(-c2ccc3c(nnn3CC3CC3)c2Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 14/20 0.44
CYP11B2 P19099 6/20 0.38
CYP11B1 P15538 5/20 0.38
CYP19A1 P11511 2/20 0.38
ADRB1 P08588 1/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3477455 0.86 GRM2 (0.48) GRM2
SCHEMBL3473809 0.82 GRM2 (0.49) GRM2CYP11B2CYP11B1
SCHEMBL3475599 0.82 GRM2 (0.46) GRM2
SCHEMBL3475600 0.81 GRM2 (0.53) GRM2CYP11B2CYP11B1
SCHEMBL3476571 0.80 GRM2 (0.53) GRM2CYP11B2CYP11B1CYP19A1
SCHEMBL3476091 0.78 GRM2 (0.40) GRM2
SCHEMBL3475603 0.77 GRM2 (0.54) GRM2
SCHEMBL3475688 0.77 GRM2 (0.49) GRM2
SCHEMBL3476498 0.76 GRM2 (0.51) GRM2
SCHEMBL3475409 0.76 GRM2 (0.53) GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO disclosed
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO disclosed