SCHEMBL3484916

SCHEMBL3484916

CCOC(=O)CNC(=O)c1ncc(-c2cccc(Cl)c2)cc1O

nearest known ligand 0.82

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 19/20 0.82
VEGFA P15692 8/20 0.82
FLT1 P17948 8/20 0.82
EGLN3 Q9H6Z9 7/20 0.82
TET3 O43151 1/20 0.72
BBOX1 O75936 1/20 0.72
ASPH Q12797 1/20 0.72
TET2 Q6N021 1/20 0.72
KDM8 Q8N371 1/20 0.72
OGFOD1 Q8N543 1/20 0.72
TET1 Q8NFU7 1/20 0.72
HIF1AN Q9NWT6 1/20 0.72
MAPT P10636 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1921387 0.90 EGLN1 (1.00) EGLN1VEGFAFLT1EGLN3TET3
SCHEMBL30239178 0.90 EGLN1 (1.00) EGLN1VEGFAFLT1EGLN3TET3
SCHEMBL1921950 0.90 EGLN1 (0.69) EGLN1VEGFAFLT1EGLN3TET3
SCHEMBL20711145 0.90 EGLN1 (0.66) EGLN1VEGFAFLT1EGLN3TET3
SCHEMBL26170368 0.89 EGLN1 (0.77) EGLN1VEGFAFLT1EGLN3TET3
SCHEMBL3485431 0.88 EGLN1 (0.72) EGLN1VEGFAFLT1EGLN3TET3
SCHEMBL23501756 0.87 EGLN1 (0.82) EGLN1VEGFAFLT1EGLN3TET3
SCHEMBL19933469 0.87 EGLN1 (0.82) EGLN1VEGFAFLT1EGLN3TET3
SCHEMBL15164149 0.85 EGLN1 (0.80) EGLN1VEGFAFLT1EGLN3TET3
SCHEMBL3484507 0.85 EGLN1 (0.60) EGLN1VEGFAFLT1EGLN3TET3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE47437-E1 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2019-06-18 US claimed
US-9598370-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2017-03-21 US claimed
US-20160009648-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE KREOS CAPITAL VII (UK) LIMITED (GB) 2016-01-14 US claimed
US-8598210-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2013-12-03 US claimed
US-20130203816-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE AKEBIA THERAPEUTICS INC. (US) 2013-08-08 US claimed
US-8343952-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS INC. (US) 2013-01-01 US claimed
US-20100331303-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE AKEBIA THERAPEUTICS, INC. 2010-12-30 US claimed
US-12612367-B2 Method for producing nitrogen-containing heteroarylcarboxamide acetic acid derivative AKEBIA THERAPEUTICS, INC. (US) 2026-04-28 US disclosed
EP-3007695-B1 COMPOSITIONS AND METHODS FOR TREATING ANEMIA AKEBIA THERAPEUTICS INC (US) 2024-02-07 EP disclosed
US-11857543-B2 Compositions and methods for treating anemia AKEBIA THERAPEUTICS, INC. (US) 2024-01-02 US disclosed
US-11857543-B2 Compositions and methods for treating anemia AKEBIA THERAPEUTICS, INC. (US) 2024-01-02 US disclosed
US-20230159462-A1 METHOD FOR PRODUCING NITROGEN-CONTAINING HETEROARYLCARBOXAMIDE ACETIC ACID DERIVATIVE KREOS CAPITAL VII (UK) LIMITED (GB) 2023-05-25 US disclosed
US-20230159462-A1 METHOD FOR PRODUCING NITROGEN-CONTAINING HETEROARYLCARBOXAMIDE ACETIC ACID DERIVATIVE KREOS CAPITAL VII (UK) LIMITED (GB) 2023-05-25 US disclosed
US-20160339005-A1 COMPOSITIONS AND METHODS FOR TREATING OCULAR DISEASES AKEBIA THERAPEUTICS, INC. (US) 2016-11-24 US disclosed
US-20160339005-A1 COMPOSITIONS AND METHODS FOR TREATING OCULAR DISEASES AKEBIA THERAPEUTICS, INC. (US) 2016-11-24 US disclosed
WO-2016161094-A1 COMPOSITIONS AND METHODS FOR TREATING ANEMIA AKEBIA THERAPEUTICS, INC. (US) 2016-10-06 WO disclosed
US-20160143891-A1 COMPOSITIONS AND METHODS FOR TREATING ANEMIA AKEBIA THERAPEUTICS, INC. (US) 2016-05-26 US disclosed
US-20160143891-A1 COMPOSITIONS AND METHODS FOR TREATING ANEMIA AKEBIA THERAPEUTICS, INC. (US) 2016-05-26 US disclosed
WO-2015112831-A1 COMPOSITIONS AND METHODS FOR TREATING OCULAR DISEASES AKEBIA THERAPEUTICS, INC. (US) 2015-07-30 WO disclosed
WO-2014200773-A2 COMPOSITIONS AND METHODS FOR TREATING ANEMIA AKEBIA THERAPEUTICS , INC. (US) 2014-12-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160143891-A1 COMPOSITIONS AND METHODS FOR TREATING ANEMIA HIF1AN, EGLN3, EGLN2 EGLN1 5/4885VEGFA 395/4885FLT1 318/4885
US-20160339005-A1 COMPOSITIONS AND METHODS FOR TREATING OCULAR DISEASES VEGFA, FLT4, AQP4 EGLN1 2391/4885VEGFA 1/4885FLT1 6/4885
US-20160009648-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, HIF1A EGLN1 6/4885VEGFA 117/4885FLT1 55/4885
US-20130203816-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, HIF1A EGLN1 6/4885VEGFA 117/4885FLT1 55/4885
US-20100331303-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, HIF1A EGLN1 6/4885VEGFA 117/4885FLT1 55/4885
US-12612367-B2 Method for producing nitrogen-containing heteroarylcarboxamide acetic acid derivative DIMT1, HIF1A, HIF1AN EGLN1 912/4885VEGFA 269/4885FLT1 2371/4885
US-20230159462-A1 METHOD FOR PRODUCING NITROGEN-CONTAINING HETEROARYLCARBOXAMIDE ACETIC ACID DERIVATIVE DIMT1, DLAT, COASY EGLN1 1247/4885VEGFA 747/4885FLT1 2745/4885
US-11857543-B2 Compositions and methods for treating anemia HIF1AN, EGLN3, EGLN2 EGLN1 5/4885VEGFA 395/4885FLT1 318/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.