SCHEMBL348853

SCHEMBL348853

NNC(=O)c1ccc(C(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.70
HDAC1 Q13547 1/20 0.70
HDAC8 Q9BY41 1/20 0.70
MPO P05164 1/20 0.53
CYP3A4 P08684 1/20 0.53
KDM5A P29375 1/20 0.53
BLM P54132 1/20 0.53
GFER P55789 1/20 0.53
PMP22 Q01453 1/20 0.53
HIF1A Q16665 1/20 0.53
MAPT P10636 4/20 0.52
ALDH1A1 P00352 3/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
OGG1 O15527 1/20 0.52
KDM4E B2RXH2 1/20 0.52
LMNA P02545 1/20 0.52
C3AR1 Q16581 1/20 0.51
CTSD P07339 1/20 0.50
AOC2 O75106 1/20 0.49
EPHX2 P34913 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31148955 0.85 HDAC6 (0.51) HDAC6HDAC1HDAC8MPOCYP3A4
SCHEMBL1771121 0.82 HDAC6 (1.00) HDAC6HDAC1HDAC8CA1CA9
SCHEMBL20078583 0.81 CYP3A4 (0.62) HDAC6HDAC1HDAC8MPOCYP3A4
Benzoic Acid Hydrazide SCHEMBL4515671 0.81 CYP3A4 (0.62) HDAC6HDAC1HDAC8MPOCYP3A4
Benzoic Acid Hydrazide SCHEMBL83514 0.81 CYP3A4 (0.62) HDAC6HDAC1HDAC8MPOCYP3A4
Benzoic Acid Hydrazide SCHEMBL1128823 0.79 CYP3A4 (0.60) HDAC6HDAC1HDAC8MPOCYP3A4
Benzoic Acid Hydrazide SCHEMBL922906 0.79 CYP3A4 (0.60) HDAC6HDAC1HDAC8MPOCYP3A4
Benzoic Acid Hydrazide SCHEMBL31087636 0.79 CYP3A4 (0.60) HDAC6HDAC1HDAC8MPOCYP3A4
Benzoic Acid Hydrazide SCHEMBL490987 0.79 CYP3A4 (0.60) HDAC6HDAC1HDAC8MPOCYP3A4
Benzoic Acid Hydrazide SCHEMBL6469726 0.79 CYP3A4 (0.60) HDAC6HDAC1HDAC8MPOCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 561 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1493747-B1 PROCESS FOR PRODUCING MODIFIED PEPTIDE DAIICHI SANKYO CO LTD (JP) 2012-12-19 EP claimed
JP-4731781-B2 2011-07-27 JP claimed
EP-2054768-A1 THERMALLY DEVELOPABLE MATERIALS CONTAINING REDUCING AGENT COMBINATIONS Carestream Health, Inc. (US) 2009-05-06 EP claimed
WO-2008048498-A1 PHOTOTHERMOGRAPHIC MATERIALS CONTAINING PRINT STABILIZERS CARESTREAM HEALTH, INC. (US) 2008-04-24 WO claimed
US-20080057450-A1 Thermally developable materials containing reducing agent combinations EASTMAN KODAK COMPANY 2008-03-06 US claimed
WO-2008024204-A1 THERMALLY DEVELOPABLE MATERIALS CONTAINING REDUCING AGENT COMBINATIONS CARESTREAM HEALTH, INC. (US) 2008-02-28 WO claimed
US-7258967-B1 Photothermographic materials containing print stabilizers CARESTREAM HEALTH, INC. (US) 2007-08-21 US claimed
EP-1257695-B1 BIOMOLECULES HAVING MULTIPLE ATTACHMENT MOIETIES FOR BINDING TO A SUBSTRATE SURFACE NANOGEN RECOGNOMICS GMBH (DE) 2007-03-07 EP claimed
EP-1191394-B1 High speed photothermographic materials and method of making and using same EASTMAN KODAK CO (US) 2006-06-14 EP claimed
JP-3638954-B2 2005-04-13 JP claimed
US-5637449-A EMULSION LAYER CONSISTS OF A PHOTOSENSITIVE SILVER HALIDE, A NON-PHOTOSENSITIVE, REDUCIBLE SILVER SOURCE, A REDUCING AGENT SYSTEM CONTAINING HINDERED PHENOL, CO-DEVELOPER, HYDROGEN ATOM DONER COMPOUND, AND A BINDER IMATION CORP (US) 1997-06-10 US claimed
WO-1997011406-A2 BLACK-AND-WHITE PHOTOTHERMOGRAFIC AND THERMOGRAFIC ELEMENTS COMPRISING AMINE COMPOUNDS AS CONTRAST ENHANCERS IMATION CORP. (US) 1997-03-27 WO claimed
WO-1997011410-A1 BLACK-AND-WHITE PHOTOTHERMOGRAPHIC AND THERMOGRAPHIC ELEMENTS COMPRISING HYDROXAMIC ACID COMPOUNDS AS CONTRAST ENHANCERS IMATION CORP. (US) 1997-03-27 WO claimed
WO-1997011407-A1 BLACK-AND-WHITE PHOTOTHERMOGRAPHIC AND THERMOGRAPHIC ELEMENTS COMPRISING HYDROGEN ATOM DONOR COMPOUNDS AS CONTRAST ENHANCERS IMATION CORP. (US) 1997-03-27 WO claimed
WO-1997011408-A1 BLACK-AND-WHITE PHOTOTHERMOGRAPHIC AND THERMOGRAPHIC ELEMENTS COMPRISING N-ACYL-HYDRAZINE COMPOUNDS AS CONTRAST ENHANCERS IMATION CORP. (US) 1997-03-27 WO claimed
US-5558983-A GRAPHIC ARTS APPLICATIONS MINNESOTA MINING & MANUFACTURING COMPANY (US) 1996-09-24 US claimed
US-5545505-A HYDROXYAMINE, ALKANOLAMINE, AND AMMONIUM PHTHLAMATE USEFUL AS CONTRAST ENHANCER WHEN USED WITH HINDERED PHENOL DEVELOPER AND TRITYL HYDRAZIDE AND/OR FORMYL-PHENYL HYDRAZIDE CO-DEVELOPER MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1996-08-13 US claimed
US-5545507-A ULTRAHIGH CONTRAST, RESOLUTION, SHARPNESS MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1996-08-13 US claimed
WO-1996021174-A2 HYDRAZIDE COMPOUNDS USEFUL AS CO-DEVELOPERS FOR BLACK-AND-WHITE PHOTOTHERMOGRAPHIC ELEMENTS MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1996-07-11 WO claimed
US-5496695-A MEDICAL DIAGNOSTIC AND GRAPHIC ARTS FILMS EXPOSED BY LASERS AND LIGHT EMITTING DIODES MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1996-03-05 US claimed