SCHEMBL3518465

SCHEMBL3518465

OC[C@H]1CCCN1Cc1nc(-c2cn(CC3CCOCC3)c3c(Cl)cccc23)ns1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 20/20 1.00
CNR2 P34972 2/20 0.54
KCNH2 Q12809 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3568197 0.86 CNR1 (1.00) CNR1CNR2KCNH2
SCHEMBL3169970 0.86 CNR1 (0.77) CNR1KCNH2
SCHEMBL3175835 0.84 CNR1 (0.85) CNR1CNR2KCNH2
SCHEMBL3188793 0.81 CNR1 (0.87) CNR1CNR2KCNH2
SCHEMBL3170037 0.80 CNR1 (1.00) CNR1CNR2KCNH2
SCHEMBL3180193 0.79 CNR1 (0.80) CNR1CNR2KCNH2
SCHEMBL3569011 0.78 CNR1 (1.00) CNR1CNR2KCNH2
SCHEMBL3570283 0.78 CNR1 (0.82) CNR1KCNH2
SCHEMBL3169302 0.77 CNR1 (0.80) CNR1CNR2KCNH2
SCHEMBL3521132 0.77 CNR1 (1.00) CNR1CNR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919471-B1 (INDOL-3-YL)-HETEROCYCLE DERIVATIVES AS AGONISTS OF THE CANNABINOID CB1 RECEPTOR MERCK SHARP & DOHME (NL) 2014-01-08 EP disclosed
US-7763732-B2 7-Chloro-3-({5-[N-(morpholin-1-ylcarboxamido)methyl]aminomethyl}-([1,2,4]-thiadiazol-3-yl))-1-(tetrahydropyran-4-yl)methyl-1H-indole, hydrochloride salt; treatment of pain N.V. ORGANON (NL) 2010-07-27 US disclosed