SCHEMBL3520359

SCHEMBL3520359

O=C(O)c1c(O)c(-c2ccccc2)cc2ncc(-c3ccccc3)nc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN3 Q9H6Z9 1/20 0.44
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
PDGFRB P09619 1/20 0.42
KDR P35968 1/20 0.42
FLT3 P36888 1/20 0.42
DHODH Q02127 2/20 0.40
TLR9 Q9NR96 1/20 0.40
PDE10A Q9Y233 1/20 0.40
BCHE P06276 1/20 0.40
PTPN1 P18031 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HPGD P15428 1/20 0.39
MAPK1 P28482 2/20 0.39
PIK3CA P42336 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3518064 0.89 SMN1; SMN2 (0.42) EGLN3NPC1RAB9ASMN1; SMN2PDGFRB
SCHEMBL3520731 0.85 SMN1; SMN2 (0.41) NPC1RAB9ASMN1; SMN2PDGFRBKDR
SCHEMBL3522312 0.83 EGLN3 (0.67) EGLN3
SCHEMBL3527577 0.79 TLR9 (0.43) NPC1RAB9ASMN1; SMN2PDGFRBKDR
SCHEMBL3525060 0.79 DHODH (0.45) EGLN3NPC1RAB9ASMN1; SMN2PDGFRB
SCHEMBL3524259 0.78 EGLN3 (0.52) EGLN3NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL3519547 0.77 KDM4E (0.42) NPC1RAB9ASMN1; SMN2DHODHPDE10A
SCHEMBL3520739 0.75 SMN1; SMN2 (0.46) NPC1RAB9ASMN1; SMN2PDGFRBKDR
SCHEMBL3520126 0.75 EGLN3 (0.62) EGLN3
SCHEMBL3519608 0.74 EGLN3 (0.58) EGLN3NPC1RAB9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100305133-A1 Prolyl Hydroxylase Inhibitors SMITHKLINE BEECHAM CORPORATION 2010-12-02 US disclosed
EP-2227770-A2 PROLYL HYDROXYLASE INHIBITORS GlaxoSmithKline LLC (US) 2010-09-15 EP disclosed
WO-2009073497-A2 PROLYL HYDROXYLASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2009-06-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100305133-A1 Prolyl Hydroxylase Inhibitors HIF1AN, EGLN3, EGLN2 EGLN3 2/4885NPC1 2674/4885RAB9A 3111/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.