SCHEMBL352396

SCHEMBL352396

Clc1cc2nc[nH]c2cc1Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.70
KDM4E B2RXH2 3/20 0.56
ALDH1A1 P00352 1/20 0.56
APEX1 P27695 1/20 0.56
RECQL P46063 1/20 0.56
BLM P54132 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
PRKCI P41743 1/20 0.47
RAD52 P43351 1/20 0.45
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
MMP12 P39900 1/20 0.42
MAPK13 O15264 1/20 0.42
CDK1 P06493 1/20 0.42
PIM1 P11309 1/20 0.42
DYRK1A Q13627 1/20 0.42
PIM3 Q86V86 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
CYP3A4 P08684 1/20 0.41
NAMPT P43490 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL22748994 0.98 MAPT (0.68) MAPTKDM4EALDH1A1APEX1RECQL
SCHEMBL14722647 0.83 MAPT (0.56) MAPTKDM4EALDH1A1APEX1RECQL
SCHEMBL31156360 0.83 MAPT (1.00) MAPTKDM4EALDH1A1APEX1RECQL
SCHEMBL30390007 0.83 MAPT (0.61) MAPTKDM4EALDH1A1APEX1RECQL
SCHEMBL29745115 0.83 MAPT (0.61) MAPTKDM4EALDH1A1APEX1RECQL
SCHEMBL23124230 0.83 MAPT (0.61) MAPTKDM4EALDH1A1APEX1RECQL
SCHEMBL3891255 0.83 MAPT (0.61) MAPTKDM4EALDH1A1APEX1RECQL
SCHEMBL2317063 0.83 MAPT (0.61) MAPTKDM4EALDH1A1APEX1RECQL
SCHEMBL3891260 0.83 MAPT (0.56) MAPTKDM4EALDH1A1APEX1RECQL
SCHEMBL30363506 0.83 MAPT (0.85) MAPTKDM4EALDH1A1APEX1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 709 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025129105-A1 COMPOSITION AND METHOD FOR DETECTION OF BIOMOLECULES VIA AROMATIC LABELING USING HETEROCYCLIC COMPOUNDS Life Technologies Corporation (US) 2025-06-19 WO claimed
US-20250199008-A1 COMPOSITION AND METHOD FOR DETECTION OF BIOMOLECULES VIA AROMATIC LABELING USING HETEROCYCLIC COMPOUNDS Life Technologies Corporation (US) 2025-06-19 US claimed
CN-120073221-A Preparation method of diaphragm for improving shock resistance of battery 扬州纳力新材料科技有限公司 2025-05-30 CN claimed
EP-3980554-B1 HYBRIDIZING ALL-LNA OLIGONUCLEOTIDES HOFFMANN LA ROCHE (CH) 2025-03-26 EP claimed
CN-118164917-A Alpha-fluoroenamine compound and preparation method and application thereof 南京工业大学 2024-06-11 CN claimed
CN-115515643-A Modified binding polypeptides for optimized drug conjugation 建新公司 2022-12-23 CN claimed
CN-107955020-B Method for synthesizing benzimidazol oxazinone compound by copper salt catalysis in one pot 西南大学 2020-09-22 CN claimed
US-20200054664-A1 METABOLIC SUPPLEMENT FORMULATION AND METHODS OF USE FOR TREATING DEPRESSION AND ANXIETY HAWKINS GERMAINE BERNARD (US) 2020-02-20 US claimed
EP-1511757-B1 NEW COMPOUNDS FOR MODULATING THE ACTIVITY OF EXCHANGE PROTEINS DIRECTLY ACTIVATED BY CAMP (EPACS) UNIV MEDISCH CENTRUM UTRECHT (NL) 2015-11-04 EP claimed
EP-2445518-A1 COBALAMIN TAXANE BIOCONJUGATES FOR TREATING EYE DISEASE Osiris Therapeutics, Inc. (US) 2012-05-02 EP claimed
EP-0701448-A4 AMPLIFICATION OF THE VITAMIN B 12? UPTAKE SYSTEM USING POLYMERS BIOTECH AUSTRALIA PTY LTD (AU) 1997-01-02 EP claimed
US-5548064-A COLONY STIMULATING FACTOR; ORAL ADMINISTERING BIOTECH AUSTRALIA PTY LIMITED (AU) 1996-08-20 US claimed
CN-1126441-A Amplification of vitamin B12 absorption System Using polymers BIOTECH AUSTRALIA PTY LTD (AU) 1996-07-10 CN claimed
CN-1126436-A Vitamin B12 mediated oral delivery systems for GCSF and EPO BIOTECH AUSTRALIA PTY LTD (AU) 1996-07-10 CN claimed
EP-0701448-A1 AMPLIFICATION OF THE VITAMIN B 12? UPTAKE SYSTEM USING POLYMERS BIOTECH AUSTRALIA PTY. LIMITED (AU) 1996-03-20 EP claimed
EP-0700295-A1 VITAMIN B 12? MEDIATED ORAL DELIVERY SYSTEMS FOR GCSF AND EPO BIOTECH AUSTRALIA PTY. LIMITED (AU) 1996-03-13 EP claimed
US-5449720-A Amplification of the VB12 uptake system using polymers BIOTECH AUSTRALIA PTY LIMITED (AU) 1995-09-12 US claimed
WO-1994027641-A1 AMPLIFICATION OF THE VITAMIN B12 UPTAKE SYSTEM USING POLYMERS BIOTECH AUSTRALIA PTY. LIMITED (AU) 1994-12-08 WO claimed
WO-1994027613-A1 VITAMIN B12 MEDIATED ORAL DELIVERY SYSTEMS FOR GCSF AND EPO BIOTECH AUSTRALIA PTY. LIMITED (AU) 1994-12-08 WO claimed
CN-1040321-A 2 ', 5 '-therapeutic use of oligomerization adenylic acid derivant UNIV TEMPLE (US) 1990-03-14 CN claimed