SCHEMBL3524919

SCHEMBL3524919

CC(C)OCCCN1C(=O)c2c(O)c(=O)c(C(=O)NCc3ccc(F)cc3)cn2CC1O

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC22A2 O15244 11/20 0.43
CYP3A4 P08684 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2187036 0.95 SLC22A2 (0.45) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL2186862 0.92 SLC22A2 (0.46) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL2187192 0.89 SLC22A2 (0.45) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL3523992 0.88 SLC22A2 (0.47) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL2242270 0.86 SLC22A2 (0.48) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL2186514 0.86 SLC22A2 (0.49) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL3526910 0.86 SLC22A2 (0.45) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL3523844 0.86 SLC22A2 (0.47) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL3522702 0.85 POU2F2 (0.44)
SCHEMBL2185152 0.85 SLC22A2 (0.45) SLC22A2CYP3A4TMEM97ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7858788-B2 Bicyclic carbamoylpyridone derivative having HIV integrase inhibitory activity SHIONOGI & CO., LTD. (JP) 2010-12-28 US disclosed