SCHEMBL3527282

SCHEMBL3527282

COc1cc2ncnc(Nc3ccc(NC(=O)c4ccccc4)cc3)c2cc1O

nearest known ligand 0.94

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 6/20 0.94
AURKA O14965 2/20 0.88
IRAK4 Q9NWZ3 1/20 0.74
MAPK14 Q16539 4/20 0.73
EGFR P00533 3/20 0.73
KDR P35968 10/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3531894 0.99 AURKB (0.92) AURKBAURKAIRAK4MAPK14EGFR
SCHEMBL3531809 0.97 AURKB (1.00) AURKBAURKAIRAK4MAPK14EGFR
Anilinoquinazoline1 SCHEMBL1066538 0.93 AURKB (1.00) AURKBAURKAIRAK4MAPK14EGFR
Anilinoquinazoline1 SCHEMBL30195580 0.93 AURKB (1.00) AURKBAURKAIRAK4MAPK14EGFR
Anilinoquinazoline1 SCHEMBL3968007 0.92 AURKB (0.98) AURKBAURKAIRAK4MAPK14EGFR
SCHEMBL8933899 0.89 AURKB (0.94) AURKBAURKAIRAK4MAPK14EGFR
Hydrochloric Acid SCHEMBL8807597 0.88 AURKB (0.92) AURKBAURKAIRAK4MAPK14EGFR
SCHEMBL5651730 0.87 AURKB (0.81) AURKBAURKAIRAK4MAPK14EGFR
SCHEMBL5239599 0.87 EGFR (0.80) AURKBAURKAIRAK4EGFRKDR
Hydrochloric Acid SCHEMBL2463942 0.86 AURKB (0.80) AURKBAURKAIRAK4MAPK14EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7709479-B1 Quinazoline derivatives and their use as pharmaceuticals ASTRAZENECA (SE) 2010-05-04 US disclosed
EP-1218354-A1 QUINAZOLINE DERIVATIVES AND THEIR USE AS PHARMACEUTICALS AstraZeneca AB (SE) 2002-07-03 EP disclosed
WO-2001021596-A1 QUINAZOLINE DERIVATIVES AND THEIR USE AS PHARMACEUTICALS ASTRAZENECA AB (SE) 2001-03-29 WO disclosed