SCHEMBL3531334

SCHEMBL3531334

Cc1ccc(S(=O)(=O)OC(=O)c2cn(-c3nc(N)c(F)cc3F)c3c(Br)c(N4CC(NC(C)C)C4)c(F)cc3c2=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47
KDM4E B2RXH2 2/20 0.32
HPGD P15428 2/20 0.32
CYP2C19 P33261 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
XBP1 P17861 1/20 0.32
NFKB1 P19838 1/20 0.32
HTT P42858 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TOP2A P11388 5/20 0.31
TOP2B Q02880 3/20 0.31
TOP1 P11387 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2919764 0.93 CYP3A4 (0.48) CYP3A4CYP2C9KDM4EHPGDCYP2C19
SCHEMBL2915542 0.90 CYP3A4 (0.51) CYP3A4CYP2C9KDM4EHPGDCYP2C19
SCHEMBL3531332 0.89 CYP3A4 (0.54) CYP3A4CYP2C9KDM4EHPGDALDH1A1
SCHEMBL2915537 0.85 CYP3A4 (0.59) CYP3A4CYP2C9KDM4EHPGDALDH1A1
SCHEMBL2918028 0.84 CYP3A4 (0.62) CYP3A4CYP2C9KDM4EHPGDALDH1A1
Hydrochloric Acid SCHEMBL2923148 0.84 CYP3A4 (0.62) CYP3A4CYP2C9KDM4EHPGDALDH1A1
SCHEMBL2922328 0.83 CYP3A4 (0.52) CYP3A4CYP2C9KDM4EHPGDCYP2C19
SCHEMBL2919763 0.82 CYP3A4 (0.55) CYP3A4CYP2C9KDM4EHPGDALDH1A1
Maleic Acid SCHEMBL2916339 0.81 CYP3A4 (0.58) CYP3A4CYP2C9KDM4EHPGDALDH1A1
Fumaric Acid SCHEMBL2916343 0.81 CYP3A4 (0.58) CYP3A4CYP2C9KDM4EHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7713997-B2 Pyridonecarboxylic acid derivatives or salts thereof WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2010-05-11 US claimed