SCHEMBL3549478

SCHEMBL3549478

NC1=NC(c2cccnc2)(c2ccc3c(c2)OCO3)c2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 8/20 0.49
CTSD P07339 5/20 0.49
BACE2 Q9Y5Z0 5/20 0.49
KCNH2 Q12809 3/20 0.47
SLC6A3 Q01959 2/20 0.40
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
GAA P10253 1/20 0.37
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
TP53 P04637 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8225744 0.91 BACE1 (0.62) BACE1CTSDBACE2KCNH2CYP11B1
SCHEMBL3548697 0.84 BACE1 (0.62) BACE1CTSDBACE2KCNH2CYP11B1
SCHEMBL2086817 0.83 BACE1 (0.43) BACE1CTSDBACE2KCNH2SLC6A3
SCHEMBL13039878 0.83 BACE1 (0.43) BACE1CTSDBACE2KCNH2SLC6A3
SCHEMBL3552663 0.83 BACE1 (0.69) BACE1CTSDBACE2KCNH2
SCHEMBL3548927 0.81 BACE1 (0.64) BACE1CTSDBACE2KCNH2
SCHEMBL3544331 0.78 BACE1 (0.51) BACE1CTSDBACE2KCNH2
SCHEMBL3559550 0.77 BACE1 (0.48) BACE1CTSDBACE2KCNH2MAPT
Trifluoroacetic Acid SCHEMBL2086300 0.77 BACE1 (0.56) BACE1CTSDBACE2KCNH2CYP11B1
SCHEMBL3549867 0.77 BACE1 (0.69) BACE1CTSDBACE2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7855213-B2 Compounds ASTRAZENECA AB (SE) 2010-12-21 US claimed