SCHEMBL3565973

SCHEMBL3565973

Cc1ccc2cc(CBr)ccc2c1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.59
CYP2A6 P11509 5/20 0.59
TDP1 Q9NUW8 1/20 0.50
ALDH1A1 P00352 2/20 0.36
NCK1 P16333 1/20 0.36
BACE1 P56817 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
IDO1 P14902 1/20 0.36
CA12 O43570 3/20 0.35
CA9 Q16790 3/20 0.35
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4312702 0.93 CYP2A6 (0.61) CYP1A2CYP2A6TDP1ALDH1A1NCK1
SCHEMBL1721014 0.85 CYP1A2 (0.44) CYP1A2CYP2A6ALDH1A1SLC6A2SLC6A3
SCHEMBL29707612 0.85 CYP1A2 (0.44) CYP1A2CYP2A6ALDH1A1SLC6A2SLC6A3
SCHEMBL14948435 0.84 CYP2A6 (0.45) CYP1A2CYP2A6TDP1SLC6A2SLC6A4
SCHEMBL10986585 0.84 CYP2A6 (0.46) CYP1A2CYP2A6TDP1ALDH1A1SLC6A2
SCHEMBL7840203 0.83 AKR1B1 (0.43) CYP1A2CYP2A6TDP1ALDH1A1KDM4E
SCHEMBL5349984 0.80 CYP1A2 (0.41) CYP1A2CYP2A6TDP1ALDH1A1SLC6A2
SCHEMBL14562409 0.79 CYP2A6 (0.50) CYP1A2CYP2A6TDP1SLC6A2SLC6A4
SCHEMBL29786773 0.79 CYP1A2 (0.64) CYP1A2CYP2A6TDP1ALDH1A1NCK1
SCHEMBL599076 0.79 CYP1A2 (0.64) CYP1A2CYP2A6TDP1ALDH1A1NCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2098527-B1 NOVEL FUSED-RING AROMATIC COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF NIPPON KAYAKU KK (JP) 2016-03-30 EP disclosed
US-8232546-B2 Fused polycyclic aromatic compound, process for producing the same, and use thereof HIROSHIMA UNIVERSITY (JP) 2012-07-31 US disclosed
US-20100065826-A1 NOVEL FUSED POLYCYCLIC AROMATIC COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2010-03-18 US disclosed
EP-2098527-A1 NOVEL FUSED-RING AROMATIC COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Hiroshima University (JP) 2009-09-09 EP disclosed
US-7579417-B2 For example, { mu-( eta 5-2-Methyl-8-phenyl-3H-cyclopenta[a]naphth-3-yl)( eta 5-2,5-dimethyldithiophenocyclopentadien-7-yl)dimethylsilanediyl]dichiorozirconium; catalyst for (co)polymerizing olefins comprising from 2 to 20 carbon atoms BASELL POLYOLEFINE GMBH (DE) 2009-08-25 US disclosed
US-7579417-B2 For example, { mu-( eta 5-2-Methyl-8-phenyl-3H-cyclopenta[a]naphth-3-yl)( eta 5-2,5-dimethyldithiophenocyclopentadien-7-yl)dimethylsilanediyl]dichiorozirconium; catalyst for (co)polymerizing olefins comprising from 2 to 20 carbon atoms BASELL POLYOLEFINE GMBH (DE) 2009-08-25 US disclosed
US-7579417-B2 For example, { mu-( eta 5-2-Methyl-8-phenyl-3H-cyclopenta[a]naphth-3-yl)( eta 5-2,5-dimethyldithiophenocyclopentadien-7-yl)dimethylsilanediyl]dichiorozirconium; catalyst for (co)polymerizing olefins comprising from 2 to 20 carbon atoms BASELL POLYOLEFINE GMBH (DE) 2009-08-25 US disclosed
EP-1697427-B1 METALLOCENE COMPOUNDS BASELL POLYOLEFINE GMBH (DE) 2008-12-24 EP disclosed
EP-1697427-B1 METALLOCENE COMPOUNDS BASELL POLYOLEFINE GMBH (DE) 2008-12-24 EP disclosed
US-20070112152-A1 Metallocene compounds BASELL POLYOLEFINE GMBH (DE) 2007-05-17 US disclosed
US-5196422-A Antiinflammatory agents, antiallergens ICI PHARMA (FR) 1993-03-23 US disclosed
US-5089513-A Antiinflammatory agents; antiallergens; asthma; side effect reduction ICI PHARMA (FR) 1992-02-18 US disclosed
US-5004744-A Durability; effectiveness at low concentration BAYER AKTIENGESELLSCHAFT (DE) 1991-04-02 US disclosed
EP-0373425-A2 Substituted pyridazinones, their preparation method and their use as insecticides BAYER AG (DE) 1990-06-20 EP disclosed
US-4513005-A SULFIDE OR SULFONE HYDROXY ACIDS LILLY INDUSTRIES LIMITED (GB) 1985-04-23 US disclosed
EP-0068739-B1 SULPHUR-CONTAINING 5-HYDROXY-ALKANOIC ACID DERIVATIVES, THEIR USE AS PHARMACEUTICAL PREPARATIONS AND PROCESS FOR THEIR PRODUCTION Lilly Industries Limited (GB) 1984-11-14 EP disclosed
EP-0068739-A1 Sulphur-containing 5-hydroxy-alkanoic acid derivatives, their use as pharmaceutical preparations and process for their production Lilly Industries Limited (GB) 1983-01-05 EP disclosed
US-4276305-A INSECTICIDES, MITICIDES HOFFMANN-LA ROCHE INC. (US) 1981-06-30 US disclosed
EP-0014455-A2 Cyclopropane(thiol)carboxylic-acid esters, processes for their preparation, pesticides containing such compounds and the use of such compounds as pesticides F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1980-08-20 EP disclosed
US-4112092-A CNS DISORDER, PARKINSON'S, CARDIOVASCULAR DISORDER SCIENCE UNION ET CIE (FR) 1978-09-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070112152-A1 Metallocene compounds NR4A2, NR4A1, NR4A3 CYP1A2 193/4885CYP2A6 1027/4885TDP1 4773/4885
US-20100065826-A1 NOVEL FUSED POLYCYCLIC AROMATIC COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF ZFX, BMX, CYP4X1 CYP1A2 615/4885CYP2A6 878/4885TDP1 4327/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.