SCHEMBL3570229

SCHEMBL3570229

Nc1ccccc1NC(=O)c1cc2ccc(CN(Cc3ccccc3)C(=O)O)cc2s1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 6/20 0.55
HDAC1 Q13547 17/20 0.50
HDAC3 O15379 3/20 0.46
NCOR2 Q9Y618 1/20 0.46
HDAC4 P56524 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3574536 0.85 HDAC2 (0.51) HDAC2HDAC1HDAC3NCOR2
SCHEMBL3565708 0.85 HDAC1 (0.71) HDAC2HDAC1HDAC3NCOR2HDAC4
SCHEMBL3571690 0.85 HDAC2 (0.48) HDAC2HDAC1HDAC3NCOR2HDAC4
SCHEMBL13074150 0.84 HDAC2 (0.61) HDAC2HDAC1HDAC3
SCHEMBL3566001 0.83 HDAC2 (0.49) HDAC2HDAC1
SCHEMBL3565292 0.83 HDAC1 (0.46) HDAC2HDAC1HDAC3NCOR2
SCHEMBL3568743 0.83 HDAC2 (0.66) HDAC2HDAC1HDAC3NCOR2HDAC4
SCHEMBL3572237 0.81 HDAC1 (0.73) HDAC2HDAC1HDAC3HDAC4HDAC7
SCHEMBL3575136 0.81 HDAC1 (0.67) HDAC2HDAC1HDAC3HDAC4HDAC7
SCHEMBL3571336 0.81 HDAC1 (0.58) HDAC2HDAC1HDAC3NCOR2HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7834034-B2 Benzothiophene derivatives MERCK SHARP & DOHME CORP. (US) 2010-11-16 US disclosed