SCHEMBL3573367

SCHEMBL3573367

CCc1cccc2c(C(N)=O)cn(CC3CCCCC3)c12

nearest known ligand 0.55

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 20/20 0.55
CNR2 P34972 5/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3169285 0.89 CNR1 (0.60) CNR1CNR2
SCHEMBL3570810 0.84 CNR1 (0.66) CNR1CNR2
SCHEMBL3520860 0.84 CNR1 (0.66) CNR1CNR2
SCHEMBL3572795 0.83 CNR1 (0.70) CNR1CNR2
SCHEMBL5562168 0.82 CNR1 (0.81) CNR1CNR2
SCHEMBL5318827 0.75 CNR1 (0.43) CNR1CNR2
SCHEMBL3576549 0.75 CNR1 (0.57) CNR1CNR2
SCHEMBL3176127 0.75 CNR1 (0.57) CNR1CNR2
SCHEMBL3518278 0.74 CNR1 (0.66) CNR1CNR2
SCHEMBL3567919 0.74 CNR1 (0.70) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7700634-B2 (Indol-3-yl) heterocycle derivatives as agonists of the cannabinoid CB1 receptor N.V. ORGANON (NL) 2010-04-20 US disclosed
CN-100522161-C (indol-3-yl) -heterocyclic derivatives as agonists of the cannabinoid CB1 receptor AKZO NOBEL NV (NL) 2009-08-05 CN disclosed
EP-1725232-B1 (INDOL-3-YL)-HETEROCYCLE DERIVATIVES AS AGONISTS OF THE CANNABINOID CB1 RECEPTOR ORGANON NV (NL) 2008-01-23 EP disclosed
US-20070142446-A1 (Indol-3-yl) heterocycle derivatives as a agonists of the cannabinoid cb1 receptor MERCK SHARP & DOHME B.V. (NL) 2007-06-21 US disclosed
CN-1929836-A (indol-3-yl) -heterocyclic derivatives as agonists of the cannabinoid CB1 receptor AKZO NOBEL NV (NL) 2007-03-14 CN disclosed
EP-1725232-A1 (INDOL-3-YL)-HETEROCYCLE DERIVATIVES AS AGONISTS OF THE CANNABINOID CB1 RECEPTOR N.V. Organon (NL) 2006-11-29 EP disclosed
WO-2005089754-A1 (INDOL-3-YL)-HETEROCYCLE DERIVATIVES AS AGONISTS OF THE CANNABINOID CB1 RECEPTOR AKZO NOBEL N.V. (NL) 2005-09-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070142446-A1 (Indol-3-yl) heterocycle derivatives as a agonists of the cannabinoid cb1 receptor CNR1, CNR2, OPRL1 CNR1 1/4885CNR2 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.