SCHEMBL3573380

SCHEMBL3573380

CC(=O)Nc1cccc(C(=O)c2ccc3c(c2)NC(=O)/C3=C/Nc2ccc(N3CCN(C)CC3)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 3/20 0.49
NTRK1 P04629 5/20 0.48
NTRK3 Q16288 2/20 0.48
NTRK2 Q16620 4/20 0.46
PRKD1 Q15139 1/20 0.43
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
CDK1 P06493 1/20 0.40
CDK4 P11802 1/20 0.40
CCNB1 P14635 1/20 0.40
CCND1 P24385 1/20 0.40
JAK3 P52333 1/20 0.40
MAP4K1 Q92918 1/20 0.40
FLT3 P36888 1/20 0.40
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3573384 1.00 CSF1R (0.49) CSF1RNTRK1NTRK3NTRK2PRKD1
SCHEMBL4757422 0.93 JAK3 (0.47) CSF1RNTRK1NTRK3NTRK2PRKD1
SCHEMBL4757425 0.93 JAK3 (0.47) CSF1RNTRK1NTRK3NTRK2PRKD1
SCHEMBL3572136 0.93 CSF1R (0.52) CSF1RNTRK1NTRK3NTRK2NPC1
SCHEMBL3572137 0.93 CSF1R (0.52) CSF1RNTRK1NTRK3NTRK2NPC1
SCHEMBL4759327 0.92 CSF1R (0.56) CSF1RNTRK1NTRK3NTRK2NPC1
SCHEMBL4757936 0.92 NPC1 (0.52) CSF1RNTRK1NTRK3NTRK2NPC1
SCHEMBL4703036 0.92 CSF1R (0.56) CSF1RNTRK1NTRK3NTRK2NPC1
SCHEMBL4757933 0.92 NPC1 (0.52) CSF1RNTRK1NTRK3NTRK2NPC1
SCHEMBL3572998 0.92 CSF1R (0.48) CSF1RNTRK3NPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902025-A1 KINASE INHIBITORS Allergan, Inc. (US) 2008-03-26 EP claimed
US-20070032478-A1 Kinase Inhibitors ALLERGAN, INC. 2007-02-08 US claimed
WO-2007008895-A1 KINASE INHIBITORS ALLERGAN, INC. (US) 2007-01-18 WO claimed
US-7749530-B2 Kinase inhibitors ALLERGAN, INC. (US) 2010-07-06 US disclosed
US-7692005-B2 Kinase inhibitors ALLERGAN, INC. (US) 2010-04-06 US disclosed
US-20090208557-A1 Kinase inhibitors ALLERGAN, INC. 2009-08-20 US disclosed
EP-1902025-A1 KINASE INHIBITORS Allergan, Inc. (US) 2008-03-26 EP disclosed
US-20070032478-A1 Kinase Inhibitors ALLERGAN, INC. 2007-02-08 US disclosed
WO-2007008895-A1 KINASE INHIBITORS ALLERGAN, INC. (US) 2007-01-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090208557-A1 Kinase inhibitors PTK2, MAP3K6, MAP3K20 CSF1R 776/4885NTRK1 307/4885NTRK3 444/4885
US-20070032478-A1 Kinase Inhibitors ABL1, LCK, ERBB2 CSF1R 877/4885NTRK1 413/4885NTRK3 418/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.