SCHEMBL358356

SCHEMBL358356

O=C(O)c1cc2cc(Br)ccc2cc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2A Q12879 2/20 0.50
GRIN2B Q13224 2/20 0.50
GRIN2C Q14957 2/20 0.50
KDM4E B2RXH2 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
POLB P06746 1/20 0.50
MAPT P10636 1/20 0.50
MCL1 Q07820 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
GRIN1 Q05586 1/20 0.50
GPR35 Q9HC97 1/20 0.50
GRIN2D O15399 1/20 0.47
GLA P06280 1/20 0.47
DHODH Q02127 1/20 0.47
RXFP1 Q9HBX9 1/20 0.46
CES2 O00748 1/20 0.46
GALR3 O60755 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31304861 1.00 GRIN2A (0.50) GRIN2AGRIN2BGRIN2CKDM4EMEN1
SCHEMBL9250304 0.98 KDM4E (0.49) GRIN2AGRIN2BGRIN2CKDM4EMEN1
Lithium Ion SCHEMBL9250300 0.82 MEN1 (0.48) KDM4EMEN1KMT2APOLBMAPT
SCHEMBL9247059 0.82 KDM4E (0.48) KDM4EMEN1KMT2APOLBMAPT
SCHEMBL5369132 0.82 GRIN2D (0.57) GRIN2AGRIN2BGRIN2CKDM4EMEN1
SCHEMBL5353853 0.82 GRIN2D (0.57) GRIN2AGRIN2BGRIN2CKDM4EMEN1
SCHEMBL29434908 0.81 CA12 (0.61) GRIN2AGRIN2BGRIN2CMEN1KMT2A
SCHEMBL124773 0.81 CA12 (0.61) GRIN2AGRIN2BGRIN2CMEN1KMT2A
SCHEMBL216334 0.81 CA12 (0.61) GRIN2AGRIN2BGRIN2CMEN1KMT2A
SCHEMBL569318 0.80 KDM4E (0.65) GRIN2AGRIN2BGRIN2CKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 149 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118184679-A Photothermal agent and preparation method thereof, photothermal nanoparticle and preparation method thereof, insulating material and self-repairing method of insulating material 中国石油天然气股份有限公司 2024-06-14 CN claimed
EP-3561003-A1 A HYBRID PIGMENT, METHOD FOR PREPARATION THEREOF AND USES THEREOF Clariant Plastics & Coatings Ltd (CH) 2019-10-30 EP claimed
JP-59076292-A None JP disclosed
WO-2025086591-A1 ROTIGOTINE PRODRUG DERIVATIVE, PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF 烟台药物研究所 2025-05-01 WO disclosed
US-20250120987-A1 METHOD FOR TREATING CANCER USING HUMAN MITOCHONDRIAL MALIC ENZYME 2 INHIBITOR NATIONAL CHUNG HSING UNIVERSITY (TW) 2025-04-17 US disclosed
US-20240424111-A1 Degrader Compounds and Uses Thereof CALICO LIFE SCIENCES LLC (US) 2024-12-26 US disclosed
CN-119176787-A Protein tyrosine phosphatase inhibitors, pharmaceutical compositions and uses thereof 艾立康药业股份有限公司 2024-12-24 CN disclosed
US-20240383886-A1 Protein Tyrosine Phosphatase Degraders and Methods of Use Thereof ABBVIE INC. 2024-11-21 US disclosed
CN-118894823-A Naphthylamide compound serving as VEGFR inhibitor and application thereof 重庆医科大学 2024-11-05 CN disclosed
CN-118184679-A Photothermal agent and preparation method thereof, photothermal nanoparticle and preparation method thereof, insulating material and self-repairing method of insulating material 中国石油天然气股份有限公司 2024-06-14 CN disclosed
EP-4359409-A1 DEGRADER COMPOUNDS AND USES THEREOF Calico Life Sciences LLC (US) 2024-05-01 EP disclosed
US-5426189-A Dopamine receptor ligands and imaging agents THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1995-06-20 US disclosed
US-5334728-A Dopamine receptor ligands and imaging agents THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1994-08-02 US disclosed
EP-0544495-A1 Improved azo pigment compositions and process for their preparation HOECHST CELANESE CORPORATION (US) 1993-06-02 EP disclosed
US-5176750-A Alkyl glycoside dispersant HOECHST CELANESE CORPORATION (US) 1993-01-05 US disclosed
US-5066695-A Plastics; heat resistance, dispersibility CIBA-GEIGY CORPORATION (US) 1991-11-19 US disclosed
JP-S5976292-A FIXING TYPE HEAT SENSITIVE MATERIAL MITSUBISHI PAPER MILLS LTD 1984-05-01 JP disclosed
US-4115055-A Mixture of water-insoluble monoazo dyestuffs for coloring textile materials consisting at least partly of linear, aromatic polyesters ROHNER AG PRATTELN (CH) 1978-09-19 US disclosed
US-4042704-A FERTILITY CONTROL AGENTS SANDOZ, INC. (US) 1977-08-16 US disclosed
US-3971741-A DISPERSION PIGMENTS BAYER AKTIENGESELLSCHAFT (DT) 1976-07-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240383886-A1 Protein Tyrosine Phosphatase Degraders and Methods of Use Thereof PTPN5, PTPN1, PTPN2 GRIN2A 4221/4885GRIN2B 4622/4885GRIN2C 3854/4885
US-20240424111-A1 Degrader Compounds and Uses Thereof PTPN1, PTPN2, PTPN5 GRIN2A 4232/4885GRIN2B 4535/4885GRIN2C 4102/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.