Formic Acid

Formic Acid

SCHEMBL3596436

Fc1ccc(-c2ccn3c(-c4cccc(Nc5ccccc5)c4)cnc3c2)cc1.O=CO

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDR P35968 15/20 0.68
FGFR3 P22607 11/20 0.68
FLT3 P36888 4/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13407717 0.94 FLT3 (0.75) KDRFGFR3FLT3
Formic Acid SCHEMBL3585405 0.93 KDR (0.65) KDRFGFR3FLT3
Formic Acid SCHEMBL3321629 0.88 FLT3 (0.85) KDRFGFR3FLT3
SCHEMBL3590857 0.86 KDR (0.66) KDRFGFR3FLT3
Formic Acid SCHEMBL3324113 0.86 KDR (0.66) KDRFGFR3FLT3
Formic Acid SCHEMBL3325020 0.86 FGFR3 (0.66) KDRFGFR3FLT3
Formic Acid SCHEMBL3323616 0.84 FGFR3 (0.73) KDRFGFR3
Formic Acid SCHEMBL3323467 0.84 FGFR3 (0.72) KDRFGFR3FLT3
Formic Acid SCHEMBL16582028 0.84 KDR (0.69) KDRFGFR3FLT3
Formic Acid SCHEMBL3323137 0.84 FGFR3 (0.71) KDRFGFR3FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121687-B1 TRICYCLIC AMINE DERIVATIVES AS PROTEIN TYROSINE KINASE INHIBITORS ASTEX THERAPEUTICS LTD (GB) 2015-10-14 EP claimed
EP-2121687-B1 TRICYCLIC AMINE DERIVATIVES AS PROTEIN TYROSINE KINASE INHIBITORS ASTEX THERAPEUTICS LTD (GB) 2015-10-14 EP disclosed
US-8513276-B2 Imidazo[1,2-a]pyridine compounds for use in treating cancer ASTEX THERAPEUTICS LIMITED (GB) 2013-08-20 US disclosed
US-20100093718-A1 Compounds ASTEX THERAPEUTICS LIMITED (GB) 2010-04-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100093718-A1 Compounds FGFR1, FGFR2, PDGFRB KDR 7/4885FGFR3 6/4885FLT3 16/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.