SCHEMBL359805

SCHEMBL359805

NS(=O)(=O)/C=C/c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PPARG P37231 6/20 0.53
LMNA P02545 2/20 0.53
NFE2L2 Q16236 2/20 0.53
PTGS2 P35354 7/20 0.51
PTGS1 P23219 6/20 0.51
PTGES2 Q9H7Z7 1/20 0.51
HSD17B10 Q99714 1/20 0.46
MAOB P27338 1/20 0.46
PKM P14618 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1205879 1.00 PPARG (0.53) PPARGLMNANFE2L2PTGS2PTGS1
SCHEMBL29175487 0.98 PPARG (0.52) PPARGLMNANFE2L2PTGS2PTGS1
SCHEMBL29026002 0.98 PPARG (0.52) PPARGLMNANFE2L2PTGS2PTGS1
SCHEMBL5766149 0.98 PPARG (0.52) PPARGLMNANFE2L2PTGS2PTGS1
SCHEMBL5766143 0.98 PPARG (0.52) PPARGLMNANFE2L2PTGS2PTGS1
SCHEMBL11539912 0.87 PTGES2 (0.50) PPARGLMNANFE2L2PTGS2PTGS1
SCHEMBL1194569 0.80 PPARG (0.57) PPARGLMNANFE2L2PTGES2MAOB
SCHEMBL19155588 0.80 PPARG (0.57) PPARGLMNANFE2L2PTGES2MAOB
SCHEMBL587895 0.80 PPARG (0.57) PPARGLMNANFE2L2PTGES2MAOB
SCHEMBL3730162 0.80 PPARG (0.57) PPARGLMNANFE2L2PTGES2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 158 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773310-B9 ALPHA, BETA-UNSATURATED SULFONES, SULFOXIDES, SULFONIMIDES, SULFINIMIDES, ACYLSULFONAMIDES AND ACYLSULFINAMIDES AND THERAPEUTIC USES THEREOF UNIV TEMPLE (US) 2012-04-25 EP claimed
EP-1773310-B1 ALPHA, BETA-UNSATURATED SULFONES, SULFOXIDES, SULFONIMIDES, SULFINIMIDES, ACYLSULFONAMIDES AND ACYLSULFINAMIDES AND THERAPEUTIC USES THEREOF UNIV TEMPLE (US) 2011-10-19 EP claimed
EP-0699191-A1 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN TEXAS BIOTECHNOLOGY CORPORATION (US) 1996-03-06 EP claimed
WO-1994027979-A1 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN IMMUNOPHARMACEUTICS, INC. (US) 1994-12-08 WO claimed
JP-58090556-A None JP disclosed
EP-3057981-B1 THERAPEUTIC CANCER VACCINE BASED ON STRESS PROTEINS RENDERED IMMUNOGENIC BRENUS PHARMA (FR) 2021-11-10 EP disclosed
US-20210207175-A1 COMPOUND FOR REGULATING GENE EDITING EFFICIENCY AND APPLICATION THEREOF SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2021-07-08 US disclosed
EP-3825409-A1 COMPOUND FOR REGULATING GENE EDITING EFFICIENCY AND APPLICATION THEREOF Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CN) 2021-05-26 EP disclosed
EP-3388425-B1 AMINOAZOLE DERIVATIVE TEIJIN PHARMA LTD (JP) 2020-08-05 EP disclosed
US-10689354-B2 Aminoazole derivative TEIJIN PHARMA LIMITED (JP) 2020-06-23 US disclosed
WO-2019238091-A1 COMPOUND FOR REGULATING GENE EDITING EFFICIENCY AND APPLICATION THEREOF 中国科学院上海有机化学研究所 2019-12-19 WO disclosed
US-10392348-B2 2-oxo-3,4-dihydroquinoline compounds as plant growth regulators SYNGENTA PARTICIPATIONS AG (CH) 2019-08-27 US disclosed
WO-1994027979-A1 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN IMMUNOPHARMACEUTICS, INC. (US) 1994-12-08 WO disclosed
EP-0467621-B1 N-phenyl-N'-alkylsulfonylureas, process for their preparation and antitumor compositions containing them LILLY CO ELI (US) 1994-06-15 EP disclosed
US-5216026-A Administering to the mammal N-1-butanesulfonamide derivatives and salts ELI LILLY AND COMPANY (US) 1993-06-01 US disclosed
EP-0467621-A1 N-phenyl-N'-alkylsulfonylureas, process for their preparation and antitumor compositions containing them ELI LILLY AND COMPANY (US) 1992-01-22 EP disclosed
JP-S5890556-A BENZAMIDE DERIVATIVE AND HERBICIDE CONTAINING THE SAME ISHIHARA SANGYO KAISHA LTD 1983-05-30 JP disclosed
US-4136180-A HYPOLIPIDEMIC SUBSTITUTED STYRENESULFONYLUREAS PFIZER INC. (US) 1979-01-23 US disclosed
US-4062960-A Hypolipidemic alkenesulfonamides PFIZER INC. (US) 1977-12-13 US disclosed
US-3983107-A ARTERIOSCLEROSIS PFIZER INC. (US) 1976-09-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10392348-B2 2-oxo-3,4-dihydroquinoline compounds as plant growth regulators CDC25B, OSR1, CDC25C PPARG 599/4885LMNA 4460/4885NFE2L2 4/4885
US-10689354-B2 Aminoazole derivative AR, NR3C2, NR5A1 PPARG 410/4885LMNA 3465/4885NFE2L2 3325/4885
US-20210207175-A1 COMPOUND FOR REGULATING GENE EDITING EFFICIENCY AND APPLICATION THEREOF TET2, ZFX, ZFR PPARG 334/4885LMNA 1544/4885NFE2L2 4073/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.