SCHEMBL3609323

SCHEMBL3609323

c1cncc(C2CCC(CCNCCC3CCC(c4cccnc4)O3)O2)c1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.69
CYP3A4 P08684 1/20 0.68
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
PTAFR P25105 1/20 0.43
SLC6A3 Q01959 1/20 0.42
CYP11B2 P19099 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13073611 0.84 CYP2A6 (0.78) CYP2A6CYP3A4SLC6A2SLC6A4PTAFR
SCHEMBL3604205 0.82 CYP2A6 (1.00) CYP2A6CYP3A4SLC6A2SLC6A4PTAFR
SCHEMBL5536201 0.82 SLC6A2 (0.62) SLC6A2SLC6A4SLC6A3
SCHEMBL13073605 0.81 CYP2A6 (0.75) CYP2A6CYP3A4SLC6A2SLC6A4PTAFR
SCHEMBL3608786 0.81 CYP2A6 (1.00) CYP2A6CYP3A4SLC6A2SLC6A4PTAFR
SCHEMBL3601299 0.81 CYP2A6 (1.00) CYP2A6CYP3A4SLC6A2SLC6A4SLC6A3
SCHEMBL3601047 0.81 CYP2A6 (1.00) CYP2A6CYP3A4SLC6A2SLC6A4PTAFR
SCHEMBL5536195 0.77 SLC6A2 (0.72) SLC6A2SLC6A4PTAFRSLC6A3
SCHEMBL13073606 0.77 CYP2A6 (0.69) CYP2A6CYP3A4SLC6A2SLC6A4PTAFR
SCHEMBL5534801 0.73 SLC6A2 (0.44) SLC6A2SLC6A4PTAFRSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2008-08-07 US claimed
WO-2005066162-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2005-07-21 WO claimed
US-8609708-B2 Synthetic compounds and derivatives as modulators of smoking or nicotine ingestion and lung cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2013-12-17 US disclosed
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2010-11-25 US disclosed
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2008-08-07 US disclosed
WO-2005066162-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2005-07-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer CYP2A13, CYP2A6, CYP2B6 CYP2A6 2/4885CYP3A4 45/4885SLC6A2 219/4885
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER CYP2A13, CYP2A6, CYP2B6 CYP2A6 2/4885CYP3A4 45/4885SLC6A2 219/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.