SCHEMBL3626552

SCHEMBL3626552

CC(C)c1ccc(-c2ccc(C(C)(c3ccc(OCc4ccccn4)cc3)C(C)C)cc2)nn1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 3/20 0.66
MAPT P10636 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MAPK14 Q16539 3/20 0.43
SMO Q99835 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ADAMTS4 O75173 1/20 0.40
SYK P43405 5/20 0.39
AURKB Q96GD4 1/20 0.39
INCENP Q9NQS7 1/20 0.39
PARP10 Q53GL7 1/20 0.39
MAOB P27338 1/20 0.38
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2999380 0.89 ALOX5AP (0.66) ALOX5APMAPTNPC1RAB9AMAPK14
SCHEMBL3000899 0.88 ALOX5AP (0.65) ALOX5APMAPTNPC1RAB9AMAPK14
SCHEMBL3000709 0.88 ALOX5AP (0.65) ALOX5APMAPTNPC1RAB9AMAPK14
SCHEMBL2989772 0.88 ALOX5AP (0.65) ALOX5APMAPTNPC1RAB9AMAPK14
SCHEMBL3003688 0.88 ALOX5AP (0.65) ALOX5APMAPTNPC1RAB9AMAPK14
SCHEMBL3002644 0.88 ALOX5AP (0.66) ALOX5APMAPTNPC1RAB9AMAPK14
SCHEMBL2997435 0.87 ALOX5AP (0.86) ALOX5APMAPTNPC1RAB9AMAPK14
SCHEMBL2993422 0.87 ALOX5AP (0.70) ALOX5APMAPTNPC1RAB9AMAPK14
SCHEMBL2991626 0.87 ALOX5AP (0.61) ALOX5APMAPK14SMOSMN1; SMN2ALDH1A1
SCHEMBL3003686 0.86 ALOX5AP (0.61) ALOX5APMAPTNPC1RAB9AMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170065-A1 DIPHENYL SUBSTITUTED ALKANES Merck Sharp & Dohme Corp. (US) 2010-04-07 EP claimed
WO-2008156721-A1 DIPHENYL SUBSTITUTED ALKANES MERCK & CO., INC. (US) 2008-12-24 WO claimed