SCHEMBL3628027

SCHEMBL3628027

CCCCN(C(=O)c1ccccn1)c1nnc(-c2cc(C)c(OC)c(C)c2)s1.CCCCN(C(=O)c1cccnc1)c1nnc(-c2cc(C)c(OC)c(C)c2)s1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 16/20 0.61
HSD17B10 Q99714 3/20 0.51
MAPT P10636 1/20 0.51
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
HPGD P15428 1/20 0.49
UBE2N P61088 1/20 0.49
NPC1 O15118 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1966885 0.93 S1PR1 (0.69) S1PR1HSD17B10MAPTKDM4EALDH1A1
SCHEMBL1969999 0.92 HSD17B10 (0.56) S1PR1HSD17B10KDM4EALDH1A1SMN1; SMN2
SCHEMBL1965848 0.85 S1PR1 (0.52) S1PR1HSD17B10KDM4EALDH1A1SMN1; SMN2
SCHEMBL1964962 0.85 S1PR1 (0.64) S1PR1HSD17B10MAPTKDM4EALDH1A1
SCHEMBL1970592 0.82 S1PR1 (0.44) S1PR1HSD17B10MAPTKDM4EALDH1A1
SCHEMBL1967851 0.80 S1PR1 (0.77) S1PR1HSD17B10KDM4EALDH1A1SMN1; SMN2
SCHEMBL1966747 0.79 S1PR1 (0.69) S1PR1HSD17B10KDM4EALDH1A1SMN1; SMN2
SCHEMBL1970812 0.79 S1PR1 (0.60) S1PR1HSD17B10KDM4EALDH1A1SMN1; SMN2
SCHEMBL1966161 0.79 S1PR1 (0.68) S1PR1HSD17B10KDM4EALDH1A1SMN1; SMN2
SCHEMBL1966359 0.79 KDM4E (0.55) S1PR1HSD17B10KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010043377-A1 NEW 2-AMIDOTHIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2010-04-22 WO disclosed