SCHEMBL3631463

SCHEMBL3631463

Cc1nc(-c2cccc(-c3cccc(S(C)(=O)=O)c3)c2)c2cccc(C(F)(F)F)c2n1.Cc1nc(-c2cccc(Br)c2)c2cccc(C(F)(F)F)c2n1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 18/20 0.55
NR1H3 Q13133 15/20 0.55
PTGS2 P35354 1/20 0.45
RXRA P19793 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3510327 0.94 NR1H2 (0.61) NR1H2NR1H3RXRA
SCHEMBL3507631 0.87 ESR1 (0.42) NR1H2PTGS2
SCHEMBL3511764 0.86 NR1H2 (0.62) NR1H2NR1H3
SCHEMBL3509019 0.83 NR1H2 (0.60) NR1H2NR1H3RXRA
SCHEMBL3505942 0.82 NR1H2 (0.64) NR1H2NR1H3RXRA
SCHEMBL3509369 0.81 NR1H2 (0.58) NR1H2NR1H3RXRA
SCHEMBL3507737 0.80 NR1H2 (0.64) NR1H2NR1H3RXRA
SCHEMBL3507401 0.80 NR1H2 (0.61) NR1H2NR1H3RXRA
SCHEMBL3505275 0.78 NR1H2 (0.55) NR1H2NR1H3RXRA
SCHEMBL3507120 0.78 NR1H2 (0.62) NR1H2NR1H3RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2142517-A2 QUINAZOLINE COMPOUNDS Wyeth (US) 2010-01-13 EP disclosed
WO-2009020683-A2 QUINAZOLINE COMPOUNDS WYETH (US) 2009-02-12 WO disclosed