SCHEMBL3633764

SCHEMBL3633764

CCCN(C(=O)Cc1cccc(C(F)(F)F)c1C(=O)O)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLQ O75417 13/20 0.53
TP53 P04637 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.40
NPC1 O15118 1/20 0.40
JAK2 O60674 1/20 0.40
RAB9A P51151 1/20 0.40
PAX8 Q06710 1/20 0.40
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
MLYCD O95822 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3633517 0.91 POLQ (0.46) POLQTP53SMN1; SMN2NPC1JAK2
SCHEMBL2149620 0.84 TP53 (0.51) POLQTP53SMN1; SMN2NPC1JAK2
SCHEMBL2148966 0.81 TP53 (0.51) TP53SMN1; SMN2NPC1JAK2RAB9A
SCHEMBL9295793 0.72 TP53 (0.62) TP53SMN1; SMN2NPC1JAK2RAB9A
SCHEMBL14230004 0.71 TP53 (0.89) TP53SMN1; SMN2NPC1JAK2RAB9A
SCHEMBL16627492 0.70 TP53 (0.70) TP53SMN1; SMN2NPC1JAK2RAB9A
SCHEMBL4757416 0.70 TP53 (0.64) TP53SMN1; SMN2NPC1JAK2RAB9A
SCHEMBL3634630 0.70 MAPT (0.38) TP53
SCHEMBL2069920 0.70 TP53 (0.68) TP53SMN1; SMN2NPC1JAK2RAB9A
SCHEMBL5480878 0.69 POLQ (0.41) POLQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2010-02-10 EP disclosed
WO-2008131779-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2008-11-06 WO disclosed