SCHEMBL3634385

SCHEMBL3634385

COc1ccc2nccc(N3CC(NC[C@H]4COC(=O)N4c4ccc5c(c4)NC(=O)CS5)C3)c2c1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.45
NCF1 P14598 1/20 0.38
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
MCHR1 Q99705 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3668033 0.89 KCNH2 (0.41) KCNH2MAOAMAOB
SCHEMBL3628040 0.87 KCNH2 (0.36) KCNH2
SCHEMBL1223133 0.86 KCNH2 (0.45) KCNH2NCF1MAOAMAOB
SCHEMBL1223135 0.86 KCNH2 (0.45) KCNH2NCF1MAOAMAOB
SCHEMBL1224241 0.81 KCNH2 (0.43) KCNH2NCF1MAOAMAOBMCHR1
SCHEMBL1224240 0.81 KCNH2 (0.43) KCNH2NCF1MAOAMAOBMCHR1
SCHEMBL1223196 0.79 KCNH2 (0.41) KCNH2NCF1MAOAMAOB
SCHEMBL3720502 0.78 KCNH2 (0.35) KCNH2
SCHEMBL3632180 0.77 KCNH2 (0.38) KCNH2
SCHEMBL3668001 0.76 DRD4 (0.40) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2144910-A2 OXAZOLIDINONE ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2010-01-20 EP disclosed
WO-2008126034-A2 OXAZOLIDINONE ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2008-10-23 WO disclosed