SCHEMBL3636302

SCHEMBL3636302

CCCc1onc(-c2c(Cl)cccc2Cl)c1COc1ccc(-c2ccc3oc(C(=O)OCC)cc(=O)c3c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 19/20 0.54
LIFR P42702 1/20 0.48
NR1I2 O75469 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
MAOB P27338 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3640853 0.94 NR1H4 (0.52) NR1H4LIFRNR1I2CYP1A2CYP3A4
SCHEMBL3639176 0.92 NR1H4 (0.64) NR1H4LIFRNR1I2CYP1A2CYP3A4
SCHEMBL2812516 0.89 NR1H4 (0.68) NR1H4LIFRNR1I2CYP1A2CYP3A4
SCHEMBL3637835 0.85 NR1H4 (0.62) NR1H4LIFRNR1I2CYP1A2CYP3A4
SCHEMBL3637820 0.84 NR1H4 (0.49) NR1H4LIFRNR1I2CYP1A2CYP3A4
SCHEMBL2814161 0.83 NR1H4 (0.65) NR1H4LIFRNR1I2CYP1A2CYP3A4
SCHEMBL3637226 0.81 NR1H4 (0.77) NR1H4LIFRNR1I2CYP1A2CYP3A4
SCHEMBL4336044 0.81 NR1H4 (0.67) NR1H4LIFRNR1I2CYP1A2CYP3A4
SCHEMBL4339399 0.81 NR1H4 (0.67) NR1H4LIFRNR1I2CYP1A2CYP3A4
SCHEMBL4337491 0.80 NR1H4 (0.65) NR1H4LIFRNR1I2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170072-A1 FARNESOID X RECEPTOR AGONISTS GlaxoSmithKline LLC (US) 2010-04-07 EP disclosed
WO-2008157270-A1 FARNESOID X RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed