Morpholine

Morpholine

SCHEMBL3637032

C1COCCN1.O=C1CNCCN1

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.52
KDM4E B2RXH2 1/20 0.52
CYP2C9 P11712 1/20 0.52
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.38
APEX1 P27695 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.33
OR51E2 Q9H255 1/20 0.31
CRBN Q96SW2 2/20 0.31
FKBP5 Q13451 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluoride SCHEMBL28311912 0.86
Piperazine SCHEMBL15224128 0.86 CRBN (0.40) GAASMN1; SMN2APEX1OR51E2CRBN
SCHEMBL29982853 0.86 CRBN (0.40) GAASMN1; SMN2APEX1OR51E2CRBN
SCHEMBL5194 0.83
SCHEMBL4393228 0.83 CRBN (0.42) GAAMEN1KMT2AOR51E2CRBN
SCHEMBL5937393 0.81
Bromide SCHEMBL28433548 0.81
Methane SCHEMBL29279661 0.81
Hydrochloric Acid SCHEMBL1583797 0.81
Charcoal, Activated SCHEMBL6719391 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2148871-A1 QUINOLINE-CARBOXAMIDE DERIVATIVES AS P2Y12 ANTAGONISTS Sanofi-Aventis (FR) 2010-02-03 EP disclosed
WO-2008128647-A1 QUINOLINE-CARBOXAMIDE DERIVATIVES AS P2Y12 ANTAGONISTS SANOFI-AVENTIS (FR) 2008-10-30 WO disclosed