SCHEMBL3637534

SCHEMBL3637534

CCCCCCOc1cccc(CCNC(C(=O)NC)C(NCCc2cccc(OCCCCC)c2)C(=O)NC)c1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 8/20 0.60
KCNH2 Q12809 2/20 0.57
CNR1 P21554 1/20 0.53
CNR2 P34972 1/20 0.53
PPARG P37231 2/20 0.52
PPARA Q07869 2/20 0.52
SMPD1 P17405 3/20 0.49
GGPS1 O95749 2/20 0.49
PLA2G4B P0C869 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3637670 0.85 CYP2D6 (0.74) CYP2D6KCNH2CNR1CNR2PPARG
SCHEMBL3014281 0.85 CYP2D6 (0.74) CYP2D6KCNH2CNR1CNR2PPARG
SCHEMBL3026768 0.85 CYP2D6 (0.74) CYP2D6KCNH2CNR1CNR2PPARG
SCHEMBL3014286 0.85 CYP2D6 (0.74) CYP2D6KCNH2CNR1CNR2PPARG
SCHEMBL3637531 0.81 CYP2D6 (0.74) CYP2D6KCNH2CNR1CNR2PPARG
SCHEMBL3022619 0.81 CYP2D6 (0.74) CYP2D6KCNH2CNR1CNR2PPARG
SCHEMBL3031673 0.79 CYP2D6 (0.73) CYP2D6KCNH2CNR1CNR2PPARG
SCHEMBL11563913 0.79 CHRM2 (0.62) CYP2D6KCNH2CNR1CNR2PPARG
SCHEMBL3635825 0.78 CYP2D6 (0.70) CYP2D6KCNH2CNR1CNR2PPARG
SCHEMBL3034043 0.77 CYP2D6 (0.76) CYP2D6KCNH2PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155663-A1 SUBSTITUTED 2- Ý2- (PHENYL) ETHYLAMINO¨ALKANEAMIDE DERIVATIVES AND THEIR USE AS SODIUM AND/OR CALCIUM CHANNEL MODULATORS Newron Pharmaceuticals S.p.A. (IT) 2010-02-24 EP disclosed
WO-2008151702-A1 SUBSTITUTED 2- [2- (PHENYL) ETHYLAMINO] ALKANEAMIDE DERIVATIVES AND THEIR USE AS SODIUM AND/OR CALCIUM CHANNEL MODULATORS NEWRON PHARMACEUTICALS S.P.A. (IT) 2008-12-18 WO disclosed