SCHEMBL363842

SCHEMBL363842

O=S(=O)(O)c1ccc(-c2ccc(C(C/C(=N\O)c3ccncc3)c3ccccc3)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.60
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 2/20 0.37
CA14 Q9ULX7 1/20 0.37
EPHX2 P34913 1/20 0.37
GSK3B P49841 5/20 0.37
ROCK1 Q13464 5/20 0.37
CLK4 Q9HAZ1 5/20 0.37
RPS6KA5 O75582 4/20 0.37
AKT1 P31749 4/20 0.37
PRKCD Q05655 4/20 0.37
PRKG2 Q13237 4/20 0.37
PRKG1 Q13976 4/20 0.37
PKN2 Q16513 4/20 0.37
GSK3A P49840 4/20 0.37
NEK4 P51957 3/20 0.37
ROCK2 O75116 3/20 0.37
MAP4K4 O95819 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363565 0.89 GPBAR1 (0.62) GPBAR1CA12CA1CA2CA9
SCHEMBL370416 0.89 GPBAR1 (0.62) GPBAR1CA12CA1CA2CA9
SCHEMBL370417 0.89 GPBAR1 (0.62) GPBAR1CA12CA1CA2CA9
SCHEMBL362642 0.88 GPBAR1 (0.61) GPBAR1CA12CA1CA2CA9
SCHEMBL369687 0.88 GPBAR1 (0.61) GPBAR1CA12CA1CA2CA9
SCHEMBL369688 0.88 GPBAR1 (0.61) GPBAR1CA12CA1CA2CA9
SCHEMBL1389598 0.86 GPBAR1 (0.58) GPBAR1EPHX2GSK3BROCK1CLK4
SCHEMBL361993 0.86 GPBAR1 (0.58) GPBAR1EPHX2GSK3BROCK1CLK4
SCHEMBL1389878 0.84 GPBAR1 (0.64) GPBAR1EPHX2GSK3BROCK1CLK4
SCHEMBL363119 0.84 GPBAR1 (0.64) GPBAR1EPHX2GSK3BROCK1CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed