SCHEMBL3638812

SCHEMBL3638812

CCCc1onc(-c2c(Cl)cccc2Cl)c1COc1ccc(-c2ccc3c(C(=O)O)cc(=O)oc3c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.56
NR1I2 O75469 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2C9 P11712 1/20 0.56
LIFR P42702 1/20 0.52
HSD17B13 Q7Z5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3637820 0.92 NR1H4 (0.49) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL3637835 0.88 NR1H4 (0.62) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL2811267 0.87 NR1H4 (0.74) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL4946841 0.85 NR1H4 (0.76) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL4950906 0.85 NR1H4 (0.75) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL4947994 0.85 NR1H4 (0.76) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL4338531 0.84 NR1H4 (0.62) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL4337362 0.84 NR1H4 (0.77) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL3637543 0.83 NR1H4 (0.77) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL3639176 0.83 NR1H4 (0.64) NR1H4NR1I2CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170072-A1 FARNESOID X RECEPTOR AGONISTS GlaxoSmithKline LLC (US) 2010-04-07 EP disclosed
WO-2008157270-A1 FARNESOID X RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed