SCHEMBL3639299

SCHEMBL3639299

Cc1nc2c(NS(=O)(=O)c3ccc(Cl)cc3Cl)c(Oc3ccc(CC(=O)O)cc3Cl)ccc2n1S(=O)(=O)c1ccc(Cl)cc1Cl

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 19/20 0.58
PTGDR Q13258 18/20 0.58
CYP3A4 P08684 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006605 0.93 PTGDR2 (0.51) PTGDR2PTGDRCYP3A4
SCHEMBL2002130 0.81 CYP3A4 (0.64) PTGDR2PTGDRCYP3A4
SCHEMBL2004052 0.73 PTGDR (1.00) PTGDR2PTGDRCYP3A4
SCHEMBL2003584 0.73 PTGDR (0.62) PTGDR2PTGDRCYP3A4
SCHEMBL2003099 0.73 PTGDR2 (0.86) PTGDR2PTGDRCYP3A4
SCHEMBL2002108 0.71 PTGDR (0.87) PTGDR2PTGDRCYP3A4
SCHEMBL4501444 0.71 PTGDR2 (0.86) PTGDR2PTGDR
SCHEMBL2001955 0.69 CYP3A4 (1.00) PTGDR2PTGDRCYP3A4
SCHEMBL2006458 0.69 PTGDR (0.60) PTGDR2PTGDRCYP3A4
SCHEMBL2009085 0.68 PTGDR (1.00) PTGDR2PTGDRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164828-A2 COMPOUNDS AS CRTH2 AND/OR PGD2 RECEPTORS MODULATORS AND THEIR USE FOR TREATING ASTHMA AND ALLERGIC INFLAMMATION Amgen Inc. (US) 2010-03-24 EP disclosed
WO-2008137027-A2 COMPOUNDS AS CRTH2 AND/OR PGD2 RECEPTORS MODULATORS AND THEIR USE FOR TREATING ASTHMA AND ALLERGIC INFLAMMATION AMGEN INC. (US) 2008-11-13 WO disclosed